SCHEMBL14560437

SCHEMBL14560437

CCCCN1C(=O)C(=O)N(Cc2ccc3ccccc3c2)C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.49
CYP1A2 P05177 2/20 0.44
CYP2A6 P11509 1/20 0.44
CTRB1 P17538 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PABPC1 P11940 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
USP2 O75604 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14560433 0.82 ELANE (0.58) CYP1A2NPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL14560436 0.77 KMT2A (0.59) KMT2AMEN1USP2POLBMAPT
SCHEMBL6968780 0.76 KMT2A (0.55) CYP1A2CTRB1RAB9AKMT2AMAPT
SCHEMBL14560545 0.76 DRD2 (0.50) NPC1RAB9ASMN1; SMN2POLBMAPT
SCHEMBL6978776 0.76 KMT2A (0.70) KMT2AMEN1MAPT
SCHEMBL14560444 0.74 CYP19A1 (0.42) AGTR1CYP1A2NPC1RAB9ASMN1; SMN2
SCHEMBL14560579 0.73 DRD2 (0.48) NPC1RAB9ASMN1; SMN2POLBMAPT
SCHEMBL2569297 0.72 PABPC1 (0.60) CYP1A2CTRB1SMN1; SMN2PABPC1ALOX15
SCHEMBL28752497 0.71 MGLL (0.61) CYP1A2CYP2A6CTRB1KMT2ADAO
SCHEMBL14560547 0.70 CDC25A (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7192967-B1 Cyclic imide-substituted pyridylalkane, alkene, alkine carboxamides useful as cytostatic and immunosuppressive agents ASTELLAS PHARMA GMBH (DE) 2007-03-20 US disclosed
US-7192967-B1 Cyclic imide-substituted pyridylalkane, alkene, alkine carboxamides useful as cytostatic and immunosuppressive agents ASTELLAS PHARMA GMBH (DE) 2007-03-20 US disclosed