SCHEMBL14680931

SCHEMBL14680931

CC(C)(C)NC(=O)C(C)(C)Cl

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
POLB P06746 2/20 0.36
APEX1 P27695 1/20 0.32
MAPK1 P28482 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
EPHX2 P34913 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474686 0.82 L3MBTL1 (0.39) EPHX1MEN1KMT2APOLBAPEX1
SCHEMBL20953659 0.75 MEN1 (0.40) EPHX1MEN1KMT2APOLBNPC1
SCHEMBL153717 0.75 L3MBTL1 (0.42) EPHX1MEN1KMT2APOLBNPC1
SCHEMBL13020558 0.74 POLB (0.36) EPHX1MEN1KMT2APOLBAPEX1
SCHEMBL18016462 0.73 ALDH1A1 (0.42) EPHX1MEN1KMT2APOLBMAPK1
SCHEMBL11831957 0.73
SCHEMBL10912920 0.72 EPHX1 (0.31) EPHX1POLB
SCHEMBL2757992 0.71 CA2 (0.48) EPHX1MEN1KMT2APOLBAPEX1
SCHEMBL11495937 0.71
SCHEMBL20852999 0.71 EPHX1 (0.37) EPHX1MEN1KMT2APOLBAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11819531-B2 Multifunctional zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2023-11-21 US disclosed
US-11819531-B2 Multifunctional zwitterionic polymer conjugates KODIAK SCIENCES INC. (US) 2023-11-21 US disclosed
US-20230277616-A9 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2023-09-07 US disclosed
US-20230277616-A9 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC. 2023-09-07 US disclosed
US-20210402015-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC (US) 2021-12-30 US disclosed
US-20200171179-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC. 2020-06-04 US disclosed
US-20170143841-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC. 2017-05-25 US disclosed
US-20170143841-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS KODIAK SCIENCES INC. 2017-05-25 US disclosed
US-20170007710-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES KODIAK SCIENCES INC. 2017-01-12 US disclosed
US-20160287715-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES KODIAK SCIENCES INC (US) 2016-10-06 US disclosed
US-20150004128-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES OLIGASIS, LLC (US) 2015-01-01 US disclosed
US-8765432-B2 Targeted drug phosphorylcholine polymer conjugates OLIGASIS, LLC (US) 2014-07-01 US disclosed
US-20140024776-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS OLIGASIS (US) 2014-01-23 US disclosed
US-20130045522-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES OLIGASIS (US) 2013-02-21 US disclosed
US-20130034517-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES OLIGASIS (US) 2013-02-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230277616-A9 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES PHOSPHO1, MSN, ZW10 EPHX1 2077/4885MEN1 1142/4885KMT2A 3850/4885
US-20160287715-A1 MULTIFUNCTIONAL ZWITTERIONIC POLYMER CONJUGATES PHOSPHO1, MSN, ZW10 EPHX1 2077/4885MEN1 1142/4885KMT2A 3850/4885
US-20130034517-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES PHOSPHO1, EPHA2, PCTP EPHX1 1170/4885MEN1 2351/4885KMT2A 2267/4885
US-20170143841-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS ACP1, PHOSPHO1, PARG EPHX1 2734/4885MEN1 3080/4885KMT2A 2142/4885
US-20170007710-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES PHOSPHO1, EPHA2, PCTP EPHX1 1170/4885MEN1 2351/4885KMT2A 2267/4885
US-20140024776-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS ACP1, PHOSPHO1, PARG EPHX1 2734/4885MEN1 3080/4885KMT2A 2142/4885
US-20200171179-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS ACP1, PHOSPHO1, PARG EPHX1 2734/4885MEN1 3080/4885KMT2A 2142/4885
US-20150004128-A1 TARGETED DRUG PHOSPHORYLCHOLINE POLYMER CONJUGATES PHOSPHO1, EPHA2, PCTP EPHX1 1170/4885MEN1 2351/4885KMT2A 2267/4885
US-11819531-B2 Multifunctional zwitterionic polymer conjugates PHOSPHO1, MSN, ZW10 EPHX1 2077/4885MEN1 1142/4885KMT2A 3850/4885
US-20210402015-A1 HIGH MOLECULAR WEIGHT ZWITTERION-CONTAINING POLYMERS ACP1, PHOSPHO1, PARG EPHX1 2734/4885MEN1 3080/4885KMT2A 2142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.