SCHEMBL1474090

SCHEMBL1474090

CCOC(=O)c1oc2ccc(O)cc2c1C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.60
KMT2A Q03164 4/20 0.60
ALDH1A1 P00352 2/20 0.60
HPGD P15428 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
HTT P42858 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
GPR55 Q9Y2T6 1/20 0.60
GAA P10253 1/20 0.57
HIF1A Q16665 5/20 0.57
PARG Q86W56 2/20 0.57
KDM4E B2RXH2 4/20 0.56
MAPT P10636 3/20 0.56
TSHR P16473 3/20 0.56
HSD17B10 Q99714 2/20 0.56
ALOX15 P16050 1/20 0.56
CASP1 P29466 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10739672 0.88 ALDH1A1 (0.70) MEN1KMT2AALDH1A1HPGDCYP1A2
SCHEMBL19661983 0.87 KCNH2 (0.66) ALDH1A1CYP1A2CYP2C9CYP2C19HIF1A
SCHEMBL754592 0.85 MEN1 (0.56) MEN1KMT2AALDH1A1HPGDCYP1A2
SCHEMBL16732898 0.84 KDM4E (0.62) MEN1KMT2AALDH1A1HTTSMN1; SMN2
SCHEMBL20893375 0.84 MAPT (0.62) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL788918 0.84 KCNH2 (0.67) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL30136795 0.84 MAPT (0.62) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2
SCHEMBL9378819 0.84 KDM4E (0.69) ALDH1A1HPGDSMN1; SMN2HIF1APARG
SCHEMBL1473247 0.83 KDM4E (0.69) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL6979902 0.83 KDM4E (0.60) MEN1KMT2AALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250275958-A1 GPCR REGULATOR AND USE THEREOF Beijing Changping Laboratory (CN) 2025-09-04 US disclosed
EP-4512803-A1 GPCR REGULATOR AND USE THEREOF Beijing Changping Laboratory (CN) 2025-02-26 EP disclosed
WO-2023202578-A1 GPCR REGULATOR AND USE THEREOF 北京昌平实验室 2023-10-26 WO disclosed
CN-116903562-A GPCR modulators and uses thereof 北京昌平实验室 2023-10-20 CN disclosed
US-20110112089-A1 Cysteine Protease Inhibitors MEDIVIR AB (SE) 2011-05-12 US disclosed
US-7915300-B2 Especially those of papain superfamily; prophylaxis or treatment of disorders stemming from misbalance of physiological proteases such as cathepsin K; (3aS,6S,6aS)-6-Fluoro-4-{(S)-4-methyl-2-[(R)-2,2,2-trifluoro-1-(4'-methanesulfonylbiphenyl-4-yl)-ethylamino]-pentanoyl}-tetrahydro-furo[3,2-b]pyrrol-3-one MEDIVIR AB (SE) 2011-03-29 US disclosed
US-20080234260-A1 Cysteine Protease inhibitors MEDIVIR AB (SE) 2008-09-25 US disclosed
WO-2005066180-A9 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB (SE) 2008-09-25 WO disclosed
WO-2007006714-A1 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB (SE) 2007-01-18 WO disclosed
WO-2007006715-A1 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB (SE) 2007-01-18 WO disclosed
EP-1701960-A1 CYSTEINE PROTEASE INHIBITORS Medivir Aktiebolag (SE) 2006-09-20 EP disclosed
WO-2005066180-A1 CYSTEINE PROTEASE INHIBITORS MEDIVIR AB (SE) 2005-07-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234260-A1 Cysteine Protease inhibitors CTSS, CTSZ, CTSK MEN1 2218/4885KMT2A 1492/4885ALDH1A1 4169/4885
US-20110112089-A1 Cysteine Protease Inhibitors CTSS, CTSZ, CTSK MEN1 2181/4885KMT2A 1689/4885ALDH1A1 4297/4885
US-20250275958-A1 GPCR REGULATOR AND USE THEREOF ARRB1, GPR3, GPR4 MEN1 3421/4885KMT2A 2867/4885ALDH1A1 2883/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.