5-Fluorouridine

5-Fluorouridine

SCHEMBL148674

O=P(O)(O)O.O=P(O)(O)O.O=P(O)(O)O.O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)cc1F

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of 5-Fluorouridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RY6 Q15077 2/20 0.68
P2RY14 Q15391 2/20 0.68
NT5E P21589 1/20 0.68
PYGM P11217 3/20 0.65
LMNA P02545 2/20 0.62
SMN1; SMN2 Q16637 2/20 0.62
TSHR P16473 1/20 0.62
MAPT P10636 1/20 0.62
PMP22 Q01453 1/20 0.62
HBB P68871 1/20 0.62
TK2 O00142 2/20 0.60
P2RY2 P41231 2/20 0.57
DNPH1 O43598 1/20 0.56
SLC28A1 O00337 1/20 0.55
SLC28A2 O43868 1/20 0.55
SLC29A1 Q99808 1/20 0.55
SLC28A3 Q9HAS3 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Fluorouridine SCHEMBL668873 1.00 P2RY6 (0.68) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL19901621 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL3385435 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL1682759 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL329381 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL12174049 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL11756887 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL17173362 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL21423048 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA
5-Fluorouridine SCHEMBL214536 0.95 PYGM (0.70) P2RY6P2RY14NT5EPYGMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 319 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2935331-B1 PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF ABBVIE INC (US) 2018-02-28 EP claimed
EP-2935331-A1 PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF AbbVie Inc. (US) 2015-10-28 EP claimed
US-20140227294-A1 PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF ABBVIE INC. (US) 2014-08-14 US claimed
WO-2014105810-A1 PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF ABBVIE INC. (US) 2014-07-03 WO claimed
US-12551570-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2026-02-17 US disclosed
US-12479927-B2 Compounds comprising cleavable linker and uses thereof INTOCELL, INC. (KR) 2025-11-25 US disclosed
US-20250186435-A1 PHARMACEUTICAL FORMULATIONS AND THEIR PREPARATIONS FOR TREATMENT OF CANCER CELLIX BIO PRIVATE LIMITED (IN) 2025-06-12 US disclosed
US-20250163159-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES ABBVIE INC (US) 2025-05-22 US disclosed
US-20250121087-A1 ANTIBODY-DRUG CONJUGATES COMPRISING ANTI-B7-H3 ANTIBODIES INTOCELL, INC. (KR) 2025-04-17 US disclosed
US-12168060-B2 Antibody-drug conjugates comprising anti-B7-H3 antibodies INTOCELL, INC. (KR) 2024-12-17 US disclosed
WO-2024187069-A1 ENGINEERING ENTEROBACTERIA TO SITE-SPECIFICALLY ACTIVATE THE ANTICANCER PRODRUG 5-FLUOROCYTOSINE FOR TREATING COLON CANCER UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-09-12 WO disclosed
CN-111378041-B Anti-EGFR antibodies and antibody drug conjugates 艾伯维公司 2024-08-02 CN disclosed
US-5736531-A ADMINISTERING TO TREAT AND PREVENT TOXICITY PRO-NEURON, INC. (US) 1998-04-07 US disclosed
EP-0831855-A1 NUCLEOTIDE ANALOGUES FOR TOPICAL TREATMENT OF PROLIFERATIVE DISEASE OF THE SKIN HOSTETLER, Karl Y. (US) 1998-04-01 EP disclosed
EP-0831849-A1 METHODS OF REDUCING TOXICITY OF CHEMOTHERAPEUTIC AND ANTIVIRAL AGENTS WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1998-04-01 EP disclosed
US-5667989-A Fungal cell wall Protein CLY4 BRISTOL-MYERS SQUIBB COMPANY (US) 1997-09-16 US disclosed
US-5654286-A Nucleotides for topical treatment of psoriasis, and methods for using same HOSTETLER KARL Y (US) 1997-08-05 US disclosed
WO-1996040165-A1 METHODS OF REDUCING TOXICITY OF CHEMOTHERAPEUTIC AND ANTIVIRAL AGENTS WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1996-12-19 WO disclosed
WO-1996040166-A1 NUCLEOTIDE ANALOGUES FOR TOPICAL TREATMENT OF PROLIFERATIVE DISEASE OF THE SKIN HOSTETLER KARL Y (US) 1996-12-19 WO disclosed
WO-1994026761-A1 TREATMENT OF CHEMOTHERAPEUTIC AGENT AND ANTIVIRAL AGENT TOXICITY WITH ACYLATED PYRIMIDINE NUCLEOSIDES PRO-NEURON, INC. (US) 1994-11-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140227294-A1 PROLACTIN RECEPTOR BINDING PROTEINS AND USES THEREOF PRLHR, LHCGR, FCGR2A P2RY6 2607/4885P2RY14 2273/4885NT5E 1158/4885
US-20250121087-A1 ANTIBODY-DRUG CONJUGATES COMPRISING ANTI-B7-H3 ANTIBODIES CD274, CD44, H1-3 P2RY6 3161/4885P2RY14 3560/4885NT5E 880/4885
US-12551570-B2 Compounds comprising cleavable linker and uses thereof FCGR2A, FCGR3B, FCGR1A P2RY6 3005/4885P2RY14 3131/4885NT5E 1008/4885
US-12168060-B2 Antibody-drug conjugates comprising anti-B7-H3 antibodies CD274, CD44, H1-3 P2RY6 3161/4885P2RY14 3560/4885NT5E 880/4885
US-12479927-B2 Compounds comprising cleavable linker and uses thereof VIP, ANTXR2, TNFRSF9 P2RY6 823/4885P2RY14 547/4885NT5E 1350/4885
US-20250163159-A1 ANTI-EGFR ANTIBODIES AND ANTIBODY DRUG CONJUGATES EGFR, ERBB2, ERBB3 P2RY6 3359/4885P2RY14 3786/4885NT5E 256/4885
US-20250186435-A1 PHARMACEUTICAL FORMULATIONS AND THEIR PREPARATIONS FOR TREATMENT OF CANCER SLC5A1, DPYD, SLC46A1 P2RY6 281/4885P2RY14 1240/4885NT5E 639/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.