SCHEMBL1491767

SCHEMBL1491767

FC(F)(F)c1ncccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 2/20 0.38
HSP90AA1 P07900 2/20 0.35
HDAC8 Q9BY41 1/20 0.35
NOS3 P29474 1/20 0.32
NOS2 P35228 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
METAP1 P53582 1/20 0.32
BLM P54132 1/20 0.32
HIF1A Q16665 1/20 0.32
DOHH Q9BU89 1/20 0.32
P4HTM Q9NXG6 1/20 0.32
TSHR P16473 1/20 0.32
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28128144 0.97 MALT1 (0.36) MALT1HSP90AA1HDAC8NOS3NOS2
Hydrochloric Acid SCHEMBL6192480 0.97 MALT1 (0.36) MALT1HSP90AA1HDAC8NOS3NOS2
Biphenyl SCHEMBL27729747 0.84 KIF11 (0.50) ALDH1A1KDM4ELMNATSHRMAPT
SCHEMBL30397418 0.84 MALT1 (0.32) MALT1
Trifluoroacetic Acid SCHEMBL38653278 0.83 L3MBTL1 (0.40) ALDH1A1KDM4ELMNABLMP4HTM
SCHEMBL30995275 0.79 MALT1 (0.34) MALT1
SCHEMBL28204675 0.78
SCHEMBL28898005 0.77 CYP2A6 (0.40) ALDH1A1CYP1A2HIF1ATSHRMAPT
Ammonia Solution, Strong SCHEMBL28127895 0.76
SCHEMBL28127892 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 810 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4688154-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - Portela & Ca., S.A. (PT) 2026-02-11 EP claimed
US-12545682-B2 Heterocyclic derivatives as P2X7 receptor antagonists BREYE THERAPEUTICS APS (DK) 2026-02-10 US claimed
CN-120040371-A Compound capable of degrading MYC in targeted manner and application thereof 中国医学科学院医药生物技术研究所 2025-05-27 CN claimed
EP-4543870-A1 NEW HETEROCYCLIC-CARBONYL-CYCLIC COMPOUNDS AS MAGL INHIBITORS F. Hoffmann-La Roche AG (CH) 2025-04-30 EP claimed
CN-119798168-A Preparation method of 5-bromo-2-trifluoromethyl pyrimidine 金凯(辽宁)生命科技股份有限公司 2025-04-11 CN claimed
WO-2025023851-A1 MORPHOLINE OREXIN RECEPTOR ANTAGONISTS BIAL - PORTELA & CA., S.A. (PT) 2025-01-30 WO claimed
US-20240425517-A1 NOVEL COMPOUND FOR DEGRADATION OF TARGET PROTEIN OR POLYPEPTIDE BY POLYUBIQUITINATION PRAZER THERAPEUTICS INC. (KR) 2024-12-26 US claimed
EP-3356387-B1 ANTIMICROBIAL POLYMYXIN DERIVATIVE COMPOUNDS UNIV MONASH (AU) 2024-06-26 EP claimed
CN-117886807-A Ferulic acid derivative containing 1,3, 4-oxadiazole and trifluoromethyl pyrimidine 贵阳学院 2024-04-16 CN claimed
WO-2024057001-A1 COMPOUNDS AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISORDERS AND CANCERS Benevolentai Cambridge Limited (GB) 2024-03-21 WO claimed
EP-2245017-A2 NOVEL HETEROCYCLES Orchid Research Laboratories Limited (IN) 2010-11-03 EP claimed
WO-2009095773-A2 NOVEL HETEROCYCLES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2009-08-06 WO claimed
US-20090118316-A1 Methods for Augmenting Bone PFZER INC. 2009-05-07 US claimed
EP-1765461-A1 PYK2 INHIBITORS FOR STIMULATION OF OSTEOBLAST FUNCTION Pharmacia & Upjohn Company LLC (US) 2007-03-28 EP claimed
WO-2005123191-A1 PYK2 INHIBITORS FOR STIMULATION OF OSTEOBLAST FUNCTION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-12-29 WO claimed
EP-1351691-A4 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA INC (US) 2005-06-22 EP claimed
WO-2004108706-A1 TRIAZOLE COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR ABBOTT GMBH & CO. KG (DE) 2004-12-16 WO claimed
EP-1351691-A1 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF Cytovia, Inc. (US) 2003-10-15 EP claimed
US-20030069239-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof CYTOVIA, INC. 2003-04-10 US claimed
WO-2002047690-A1 SUBSTITUTED 2-ARYL-4-ARYLAMINOPYRIMIDINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2002-06-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240425517-A1 NOVEL COMPOUND FOR DEGRADATION OF TARGET PROTEIN OR POLYPEPTIDE BY POLYUBIQUITINATION ADRM1, SUMO1, SUMO2 MALT1 3231/4885HSP90AA1 789/4885HDAC8 1381/4885
US-20090118316-A1 Methods for Augmenting Bone PTK2, PHKA2, BMP2K MALT1 4682/4885HSP90AA1 3476/4885HDAC8 4006/4885
US-20030069239-A1 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof API5, CASP2, APAF1 MALT1 291/4885HSP90AA1 1802/4885HDAC8 467/4885
US-12545682-B2 Heterocyclic derivatives as P2X7 receptor antagonists P2RX7, P2RX3, P2RX1 MALT1 2880/4885HSP90AA1 3958/4885HDAC8 2824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.