SCHEMBL15436231

SCHEMBL15436231

Cc1ccc(-c2c(C(=O)OC(C)(C)C)ccnc2NCc2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.42
BDKRB1 P46663 5/20 0.42
PSMB1 P20618 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
HPGD P15428 2/20 0.41
KDR P35968 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ASPH Q12797 1/20 0.40
KDM8 Q8N371 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CDC7 O00311 1/20 0.39
DBF4 Q9UBU7 1/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15436232 0.76 NOS2 (0.43) ACHENPSR1HPGDKDM4ESMN1; SMN2
SCHEMBL451920 0.70 PTGS2 (0.45) ACHENPSR1HPGDKDM4EALDH1A1
SCHEMBL4220977 0.69 CDC7 (0.56) HPGDKDM5BKDM4ECDC7ALDH1A1
SCHEMBL3291794 0.68 CA1 (0.53) HPGDKDM4EALDH1A1LMNAGAA
SCHEMBL5871444 0.67 PKM (0.58) BDKRB1HPGDKDRKDM5BKDM4E
SCHEMBL2087990 0.66 HTT (0.65) NPSR1KDRKDM4ESMN1; SMN2CDC7
SCHEMBL27808272 0.66 IDO1 (0.51) KDM4ESMN1; SMN2ALDH1A1GAAMAPT
SCHEMBL16625628 0.66 KDR (0.84) KDRKDM4EALDH1A1LMNAGAA
SCHEMBL16989282 0.66 KLKB1 (0.46) BDKRB1KDM4EASPHKDM8ALDH1A1
SCHEMBL517 0.66 SLC6A3 (0.50) ACHESMN1; SMN2ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410857-B1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK SHARP & DOHME (US) 2014-01-29 EP disclosed