SCHEMBL15436232

SCHEMBL15436232

Cc1ccc(-c2cnc(NCc3ccccc3)cc2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.43
CCNT1 O60563 1/20 0.42
ACHE P22303 1/20 0.41
EED O75530 1/20 0.41
ALDH1A1 P00352 5/20 0.40
LMNA P02545 2/20 0.40
RAB9A P51151 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTT P42858 1/20 0.40
CYP1A2 P05177 5/20 0.40
CYP2D6 P10635 3/20 0.40
HSD17B10 Q99714 3/20 0.40
CLK4 Q9HAZ1 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MAPK1 P28482 4/20 0.39
CYP3A4 P08684 3/20 0.39
TP53 P04637 2/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15436231 0.76 ACHE (0.42) ACHEALDH1A1LMNARAB9ANPSR1
SCHEMBL451920 0.76 PTGS2 (0.45) ACHEALDH1A1LMNANPSR1HTT
SCHEMBL2487626 0.73 CYP46A1 (0.51) ALDH1A1LMNAHSD17B10MAPK1MAPT
SCHEMBL4220977 0.71 CDC7 (0.56) ALDH1A1LMNACLK4MAPTHPGD
SCHEMBL517 0.70 SLC6A3 (0.50) ACHEALDH1A1LMNARAB9ACYP1A2
SCHEMBL3291794 0.69 CA1 (0.53) ALDH1A1LMNARAB9AHTTMAPT
SCHEMBL9709560 0.68 CD38 (0.50) RAB9AHTTSMN1; SMN2KDM4EMEN1
SCHEMBL27791830 0.68 CYP2C19 (0.47) RAB9AHTTSMN1; SMN2KDM4EMEN1
SCHEMBL1069726 0.66 FOLH1 (0.47) ACHEALDH1A1MEN1KMT2A
SCHEMBL4220608 0.66 ADRA1A (0.46) ALDH1A1HSD17B10CLK4HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410857-B1 P2X3, RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK SHARP & DOHME (US) 2014-01-29 EP disclosed