SCHEMBL15443081

SCHEMBL15443081

Cc1cn(-c2ccc3[nH]c(-c4ccc(C)c(C#Cc5cnc6cccnn56)c4)nc3c2)cn1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 11/20 0.51
DDR1 Q08345 1/20 0.43
CSF1R P07333 1/20 0.41
ROR1 Q01973 7/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15443267 0.94 ABL1 (0.51) ABL1DDR1CSF1RROR1
SCHEMBL16644546 0.83 ABL1 (0.53) ABL1DDR1CSF1RROR1
SCHEMBL20144337 0.75 NPBWR1 (0.44)
SCHEMBL15443243 0.73 ABL1 (0.58) ABL1DDR1CSF1R
SCHEMBL15445593 0.73 MAOA (0.41)
SCHEMBL25649582 0.69 ABL1 (0.56) ABL1DDR1CSF1RROR1
SCHEMBL14705592 0.68 CSF1R (0.55) ABL1DDR1CSF1RROR1
SCHEMBL17471717 0.68 CSF1R (0.57) ABL1CSF1RROR1
SCHEMBL16283150 0.67 NPC1 (0.44)
SCHEMBL16644581 0.67 ABL1 (1.00) ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3186247-B1 PROTEIN KINASE INHIBITORS ASTAR BIOTECH LLC (US) 2021-03-03 EP disclosed
EP-2880038-B1 PROTEIN KINASE INHIBITORS ASTAR BIOTECH LLC (US) 2018-05-16 EP disclosed
US-9174996-B2 Protein kinase inhibitors ASTAR BIOTECH LLC (US) 2015-11-03 US disclosed
US-20140364436-A1 Protein Kinase Inhibitors ASTAR BIOTECH LLC (US) 2014-12-11 US disclosed
US-8859553-B2 Protein kinase inhibitors ASTAR BIOTECH LLC (US) 2014-10-14 US disclosed
US-20140031354-A1 Protein Kinase Inhibitors ASTAR BIOTECH LLC (US) 2014-01-30 US disclosed
US-20070004635-A1 Method of treating interferon non-responders using HCV protease inhibitor SCHERING CORPORATION 2007-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070004635-A1 Method of treating interferon non-responders using HCV protease inhibitor IFNAR1, IFNG, IRF3 ABL1 566/4885DDR1 4558/4885CSF1R 2852/4885
US-20140364436-A1 Protein Kinase Inhibitors MAP3K9, MAP3K6, MAP3K8 ABL1 171/4885DDR1 1861/4885CSF1R 2152/4885
US-20140031354-A1 Protein Kinase Inhibitors MAP3K1, MAP3K5, MAP3K7 ABL1 134/4885DDR1 1414/4885CSF1R 1954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.