SCHEMBL20144337

SCHEMBL20144337

Cc1cn(-c2ccc3[nH]c(-c4ccc(C)c(C)c4)nc3c2)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.44
MAOA P21397 4/20 0.43
MAOB P27338 4/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
PKM P14618 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15445593 0.90 MAOA (0.41) NPBWR1MAOAMAOBNPC1RAB9A
SCHEMBL16283150 0.83 NPC1 (0.44) MAOAMAOBNPC1RAB9APKM
SCHEMBL15442436 0.80 MAOA (0.43) NPBWR1MAOAMAOBNPC1RAB9A
SCHEMBL15443081 0.75 ABL1 (0.51)
SCHEMBL23049050 0.74 NPBWR1 (0.42) NPBWR1NPC1RAB9APKMSMN1; SMN2
SCHEMBL12347958 0.69 NPC1 (0.68) NPBWR1NPC1RAB9APKMSMN1; SMN2
SCHEMBL29848567 0.69 NR2E1 (0.61) NPBWR1PSEN1PSEN2APH1BNCSTN
SCHEMBL13533794 0.69 NPC1 (0.60) NPBWR1NPC1RAB9APKMSMN1; SMN2
SCHEMBL21976216 0.67 ALOX5 (0.65) NPBWR1NPC1RAB9APKMSMN1; SMN2
Hydrochloric Acid SCHEMBL7279599 0.67 ALDH1A1 (0.51) NPBWR1NPC1RAB9APKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2880038-B1 PROTEIN KINASE INHIBITORS ASTAR BIOTECH LLC (US) 2018-05-16 EP disclosed