SCHEMBL15475873

SCHEMBL15475873

OB(O)c1c(O)cccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.39
ALDH1A1 P00352 2/20 0.38
EGFR P00533 2/20 0.38
CA2 P00918 2/20 0.38
LMNA P02545 2/20 0.38
FYN P06241 2/20 0.38
MMP9 P14780 2/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 2/20 0.38
RECQL P46063 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
ADAMTS4 O75173 1/20 0.38
CA1 P00915 1/20 0.38
MMP2 P08253 1/20 0.38
MMP8 P22894 1/20 0.38
CA6 P23280 1/20 0.38
CDK2 P24941 1/20 0.38
MMP12 P39900 1/20 0.38
ADAMTS5 Q9UNA0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29469044 1.00 ERN1 (0.39) ERN1ALDH1A1EGFRCA2LMNA
SCHEMBL146988 0.85 CES2 (0.42) ERN1CA6CES2CES1CA4
SCHEMBL3784650 0.82 ALOX15 (0.47) ERN1ALDH1A1EGFRCA2LMNA
SCHEMBL25725600 0.81 ERN1 (0.39) ERN1ALDH1A1EGFRCA2LMNA
SCHEMBL9893710 0.76 CES2 (0.36) ERN1CES2CES1KDM4EALB
Magnesium Chloride Anhydrous SCHEMBL20694920 0.76 CES2 (0.36) ERN1ALDH1A1ALOX15CES2CES1
SCHEMBL29427089 0.74 ACHE (0.48) ERN1ALDH1A1CA2CA1CES2
SCHEMBL29469267 0.74 GAA (0.42) LMNAHPGDCES2CES1KDM4E
SCHEMBL321378 0.74 GAA (0.42) LMNAHPGDCES2CES1KDM4E
SCHEMBL6007162 0.74 ACHE (0.48) ERN1ALDH1A1CA2CA1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 456 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116731315-B Boron-containing phthalonitrile resin and preparation method and application thereof 中国科学院化学研究所 2024-06-21 CN claimed
CN-118184818-A Functionalized high molecular polymer, visualized embolism microsphere prepared by microfluidic technology and application 四川大学 2024-06-14 CN claimed
CN-116731315-A Boron-containing phthalonitrile resin and preparation method and application thereof 中国科学院化学研究所 2023-09-12 CN claimed
CN-111217843-B Method for synthesizing 2-fluoro-6-hydroxyphenylboronic acid 大连联化化学有限公司 2022-07-01 CN claimed
CN-111217843-A Method for synthesizing 2-fluoro-6-hydroxyphenylboronic acid 大连联化化学有限公司 2020-06-02 CN claimed
US-12630547-B2 RAS protein degraders, pharmaceutical compositions thereof, and their therapeutic applications BIOTHERYX, INC. (US) 2026-05-19 US disclosed
US-12630566-B2 KRas G12D inhibitors Mirati Therapeutics, Inc. (US) 2026-05-19 US disclosed
CN-116829557-B Pentaheterocycle compound, preparation method and application thereof 上海艾力斯医药科技股份有限公司 2026-05-12 CN disclosed
EP-4234546-B1 IMPROVED SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND AMGEN INC (US) 2026-04-15 EP disclosed
US-12594275-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-04-07 US disclosed
US-12582657-B2 Combination therapy including a KRAS G12C inhibitor and one or more additional pharmaceutically active agents for the treatment of cancers AMGEN INC. (US) 2026-03-24 US disclosed
US-12558356-B2 Immunophilin binding agents and uses thereof THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2026-02-24 US disclosed
US-20160024077-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK (NO. 5) LIMITED (GB) 2016-01-28 US disclosed
EP-2970274-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION Bristol-Myers Squibb Company (US) 2016-01-20 EP disclosed
US-9079903-B2 Heterocyclic compound and organic light-emitting device including the same SAMSUNG DISPLAY CO., LTD. (KR) 2015-07-14 US disclosed
EP-2888266-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION Bristol-Myers Squibb Company (US) 2015-07-01 EP disclosed
US-8906929-B2 Inhibitors of human immunodeficiency virus replication BRISTOL-MYERS SQUIBB COMPANY (US) 2014-12-09 US disclosed
WO-2014159959-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2014-10-02 WO disclosed
US-20140051692-A1 Inhibitors of Human Immunodeficiency Virus Replication VIIV HEALTHCARE UK (NO. 5) LIMITED (GB) 2014-02-20 US disclosed
WO-2014028384-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2014-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12630547-B2 RAS protein degraders, pharmaceutical compositions thereof, and their therapeutic applications KRAS, RSU1, NRAS ERN1 1120/4885ALDH1A1 3991/4885EGFR 479/4885
US-12594275-B2 Immunophilin binding agents and uses thereof CCR1, CCRL2, CCR3 ERN1 3013/4885ALDH1A1 3009/4885EGFR 2717/4885
US-12630566-B2 KRas G12D inhibitors KRAS, NRAS, HRAS ERN1 2008/4885ALDH1A1 1816/4885EGFR 117/4885
US-12582657-B2 Combination therapy including a KRAS G12C inhibitor and one or more additional pharmaceutically active agents for the treatment of cancers KRAS, NRAS, BRAF ERN1 3092/4885ALDH1A1 1774/4885EGFR 10/4885
US-12558356-B2 Immunophilin binding agents and uses thereof CCRL2, CFB, CCR3 ERN1 4095/4885ALDH1A1 2201/4885EGFR 1974/4885
US-20160024077-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION EIF2AK2, RTF2, MAVS ERN1 428/4885ALDH1A1 3508/4885EGFR 3789/4885
US-20140051692-A1 Inhibitors of Human Immunodeficiency Virus Replication EIF2AK2, RTF2, MAVS ERN1 289/4885ALDH1A1 3327/4885EGFR 3735/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.