SCHEMBL15544868

SCHEMBL15544868

O=C(C1CNc2cc(F)cc(F)c21)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
P2RX7 Q99572 3/20 0.35
ALDH1A1 P00352 6/20 0.34
POLB P06746 1/20 0.34
CNR2 P34972 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.32
GRM1 Q13255 1/20 0.31
ENPP3 O14638 1/20 0.31
CA12 O43570 1/20 0.31
ENPP1 P22413 1/20 0.31
ENPP2 Q13822 1/20 0.31
CA9 Q16790 1/20 0.31
HSD11B1 P28845 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545602 0.78 ALDH1A1 (0.35) KCNQ3KCNQ2P2RX7ALDH1A1POLB
SCHEMBL15544370 0.76 CNR2 (0.41) KCNQ3KCNQ2P2RX7ALDH1A1CNR2
SCHEMBL15545632 0.71 P2RX7 (0.41) P2RX7ALDH1A1CNR2SMN1; SMN2NPSR1
SCHEMBL15545467 0.70 KCNH2 (0.41) P2RX7ALDH1A1CNR2
SCHEMBL15544668 0.69 ALDH1A1 (0.43) P2RX7ALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL15544852 0.69 LMNA (0.43) P2RX7ALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL15545052 0.68 P2RX4 (0.39) P2RX7ALDH1A1POLBCNR2LMNA
SCHEMBL15545277 0.68 SMN1; SMN2 (0.47) KCNQ3KCNQ2P2RX7CNR2SMN1; SMN2
SCHEMBL15545879 0.65 ALDH1A1 (0.44) P2RX7ALDH1A1POLBSMN1; SMN2NPSR1
SCHEMBL15544368 0.65 ALDH1A1 (0.44) P2RX7ALDH1A1POLBSMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870139-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
WO-2014005968-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed