SCHEMBL15545182

SCHEMBL15545182

O=C1C2CC3CC1CC(C(=O)C1CNc4ccccc41)(C3)C2

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.42
ALDH1A1 P00352 4/20 0.38
CNR2 P34972 3/20 0.35
IDH1 O75874 1/20 0.35
EPHX2 P34913 1/20 0.35
CYP17A1 P05093 2/20 0.33
CYP19A1 P11511 2/20 0.33
KDM4E B2RXH2 2/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
PRMT5 O14744 1/20 0.32
WDR77 Q9BQA1 1/20 0.32
GRM5 P41594 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545467 0.90 KCNH2 (0.41) KCNH2ALDH1A1CNR2IDH1CYP17A1
SCHEMBL15546001 0.78 SMN1; SMN2 (0.46) KCNH2ALDH1A1CNR2KDM4ETSHR
SCHEMBL15544668 0.73 ALDH1A1 (0.43) ALDH1A1EPHX2CYP17A1CYP19A1KDM4E
SCHEMBL15544852 0.73 LMNA (0.43) ALDH1A1EPHX2CYP17A1CYP19A1KDM4E
SCHEMBL15544370 0.72 CNR2 (0.41) ALDH1A1CNR2CYP17A1CYP19A1TSHR
SCHEMBL15545052 0.72 P2RX4 (0.39) ALDH1A1CNR2CYP17A1CYP19A1KDM4E
SCHEMBL15544373 0.70 FAAH (0.48) ALDH1A1CNR2EPHX2KDM4ETSHR
SCHEMBL27862075 0.70 ALDH1A1 (0.46) KCNH2ALDH1A1EPHX2PRMT5WDR77
SCHEMBL15545061 0.69 P2RX7 (0.41) ALDH1A1CNR2EPHX2LMNA
SCHEMBL15545632 0.69 P2RX7 (0.41) ALDH1A1CNR2IDH1EPHX2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2870139-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. Hoffmann-La Roche AG (CH) 2015-05-13 EP disclosed
WO-2014005968-A1 NOVEL ADAMANTYL DERIVATIVES AS CANNABINOID RECEPTOR 2 AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2014-01-09 WO disclosed