SCHEMBL15569271

SCHEMBL15569271

C=Cc1c(Cl)cc(C)cc1C#N

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.33
GABRG2 P18507 2/20 0.33
GABRB3 P28472 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
GABRB2 P47870 1/20 0.33
PGK1 P00558 1/20 0.33
TRPV4 Q9HBA0 1/20 0.32
AR P10275 1/20 0.30
SLC22A12 Q96S37 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL589904 0.80 TP53 (0.34) ALDH1A1HPGD
SCHEMBL19431432 0.76 L3MBTL1 (0.33) ALDH1A1KDM4EGAA
SCHEMBL15958850 0.74 TRPV4 (0.38) GABRA1GABRG2GABRB3ALDH1A1KDM4E
SCHEMBL15322142 0.70 AR (0.37) ALDH1A1AR
SCHEMBL26457742 0.69 ALDH1A1 (0.35) GABRA1GABRG2GABRB3ALDH1A1KDM4E
SCHEMBL11852191 0.67 GABRA1 (0.44) GABRA1GABRG2GABRB3ALDH1A1HPGD
SCHEMBL6416771 0.66 ALDH1A1 (0.38) GABRA1GABRG2GABRB3ALDH1A1KDM4E
SCHEMBL410587 0.66 TRPV4 (0.57) GABRA1GABRG2GABRB3ALDH1A1KDM4E
SCHEMBL27974294 0.66 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDAR
SCHEMBL366053 0.66 VCAM1 (0.48) GABRA1GABRG2GABRB3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013149996-A9 SUBSTITUTED TRICYCLIC COMPOUNDS WITH ACTIVITY TOWARDS EP1 RECEPTORS ALMIRALL, S.A. (ES) 2014-02-20 WO disclosed