SCHEMBL15747222

SCHEMBL15747222

COP(=O)(OC[C@H]1O[C@@H](n2cnc3c(=O)[nH]c(N)nc32)[C@@H](O)C1O)OP(=O)(O)OP(=O)(O)O

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.71
TGM2 P21980 1/20 0.70
FUT5 Q11128 1/20 0.65
IMPDH2 P12268 5/20 0.65
IMPDH1 P20839 1/20 0.65
KRAS P01116 4/20 0.64
HINT1 P49773 1/20 0.61
TAS1R3 Q7RTX0 1/20 0.60
TAS1R1 Q7RTX1 1/20 0.60
P2RY6 Q15077 2/20 0.60
P2RY2 P41231 1/20 0.60
P2RY4 P51582 1/20 0.60
ENPP1 P22413 2/20 0.59
P2RY1 P47900 2/20 0.59
P2RY12 Q9H244 1/20 0.59
DCPS Q96C86 1/20 0.59
P2RX3 P56373 2/20 0.59
P2RX1 P51575 1/20 0.59
P2RY11 Q96G91 1/20 0.59
P2RX4 Q99571 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20850061 1.00 NT5E (0.71) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL28165608 1.00 NT5E (0.71) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL18648315 1.00 NT5E (0.71) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL28275952 0.95 NT5E (0.75) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL21413213 0.94 NT5E (0.70) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL27819299 0.94 NT5E (0.74) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL28222628 0.94 NT5E (0.74) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL8501729 0.94 NT5E (0.74) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL574773 0.94 NT5E (0.74) NT5ETGM2FUT5IMPDH2IMPDH1
SCHEMBL4366555 0.93 NT5E (0.73) NT5ETGM2FUT5IMPDH2IMPDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751925-B2 Alternative nucleic acid molecules containing reduced uracil content and uses thereof MODERNATX, INC. (US) 2017-09-05 US disclosed
US-20170175129-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2017-06-22 US disclosed
US-20170136131-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF Modema Therapeutics, Inc. (US) 2017-05-18 US disclosed
US-20170136132-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. (US) 2017-05-18 US disclosed
US-9597380-B2 Terminally modified RNA MODERNATX, INC. (US) 2017-03-21 US disclosed
US-20160354493-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNATX, INC. 2016-12-08 US disclosed
US-20160354490-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2016-12-08 US disclosed
US-20160354491-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2016-12-08 US disclosed
US-20160354492-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2016-12-08 US disclosed
US-20160348099-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS INC (US) 2016-12-01 US disclosed
US-20160304552-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. 2016-10-20 US disclosed
US-20160264614-A1 POLYNUCLEOTIDE MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. (US) 2016-09-15 US disclosed
US-20160237108-A1 POLYNUCLEOTIDE MOLECULES AND USES THEREOF ARES CAPITAL CORPORATION, AS AGENT 2016-08-18 US disclosed
US-20160237134-A1 ALTERNATIVE NUCLEIC ACID MOLECULES CONTAINING REDUCED URACIL CONTENT AND USES THEREOF ARES CAPITAL CORPORATION, AS AGENT 2016-08-18 US disclosed
US-20150307542-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF MODERNATX, INC. 2015-10-29 US disclosed
US-20150167017-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF MODERNA THERAPEUTICS, INC. 2015-06-18 US disclosed
US-20140147454-A1 TERMINALLY MODIFIED RNA MODERNA THERAPEUTICS, INC. (US) 2014-05-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (14 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160354492-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20160264614-A1 POLYNUCLEOTIDE MOLECULES AND USES THEREOF POLRMT, POLN, NSUN3 NT5E 35/4885TGM2 2867/4885FUT5 1345/4885
US-20160304552-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20160348099-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20170136132-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, RNGTT, NSUN3 NT5E 67/4885TGM2 2234/4885FUT5 2056/4885
US-20160354490-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20160237134-A1 ALTERNATIVE NUCLEIC ACID MOLECULES CONTAINING REDUCED URACIL CONTENT AND USES THEREOF RNMT, NSUN2, ADAR NT5E 152/4885TGM2 1926/4885FUT5 1862/4885
US-20160354491-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20170175129-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, RNGTT, NSUN3 NT5E 67/4885TGM2 2234/4885FUT5 2056/4885
US-20170136131-A1 ALTERNATIVE NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, RNGTT, NSUN3 NT5E 67/4885TGM2 2234/4885FUT5 2056/4885
US-20160354493-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20140147454-A1 TERMINALLY MODIFIED RNA RNGTT, NSUN3, RNMT NT5E 234/4885TGM2 3781/4885FUT5 641/4885
US-20150307542-A1 MODIFIED NUCLEIC ACID MOLECULES AND USES THEREOF NSUN2, ADAR, NSUN3 NT5E 32/4885TGM2 1916/4885FUT5 1042/4885
US-20160237108-A1 POLYNUCLEOTIDE MOLECULES AND USES THEREOF NSUN3, POLRMT, TRDMT1 NT5E 97/4885TGM2 2945/4885FUT5 261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.