SCHEMBL15775763

SCHEMBL15775763

COc1nc(-c2ccc(C#N)cc2)cc2c(N)cccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SQOR Q9Y6N5 11/20 0.49
ACP1 P24666 3/20 0.45
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2C P18825 1/20 0.39
HTR1D P28221 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR7 P34969 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775442 0.89 SQOR (0.48) SQORACP1ALDH1A1MEN1KMT2A
SCHEMBL15775748 0.84 SQOR (0.53) SQORACP1KDM4EALDH1A1
SCHEMBL15775389 0.83 ESR1 (0.45) SQORKDM4EALDH1A1NPC1MAPT
SCHEMBL13443755 0.81 SQOR (0.57) SQORACP1KDM4EALDH1A1NPC1
SCHEMBL15775312 0.80 SQOR (0.44) SQORACP1KDM4EALDH1A1NPC1
SCHEMBL15775248 0.80 PARP1 (0.47) SQORACP1KDM4ENPC1MAPT
SCHEMBL15775799 0.77 SQOR (0.54) SQORKDM4EALDH1A1GAAMAPT
SCHEMBL15775605 0.76 NR1I3 (0.53) SQOR
SCHEMBL15775546 0.73 XDH (0.47) SQORKDM4EALDH1A1GAA
SCHEMBL15775195 0.73 HSP90AA1 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed