SCHEMBL15775799

SCHEMBL15775799

COc1cccc(-c2cc3c(N)cccc3c(OC)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SQOR Q9Y6N5 1/20 0.54
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
VDR P11473 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
AHR P35869 1/20 0.52
NR1I3 Q14994 1/20 0.52
ADORA2A P29274 2/20 0.48
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MKNK1 Q9BUB5 1/20 0.45
MKNK2 Q9HBH9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775605 0.85 NR1I3 (0.53) SQORNR1I3MAP4K4TLR8
SCHEMBL15775748 0.82 SQOR (0.53) SQORKDM4EALDH1A1HPGDSYK
SCHEMBL15775546 0.82 XDH (0.47) SQORKDM4EALDH1A1HPGDGAA
SCHEMBL15775442 0.82 SQOR (0.48) SQORCYP1A2CYP3A4CYP2C9ADORA2A
SCHEMBL15775389 0.81 ESR1 (0.45) SQORCYP1A2CYP3A4CYP2C9ADORA2A
SCHEMBL21586163 0.80 MAP4K4 (0.56) SQORCYP1A2CYP3A4VDRCYP2C9
SCHEMBL15775590 0.78 NPC1 (0.49) SQORCYP1A2CYP3A4VDRCYP2C9
SCHEMBL15775248 0.77 PARP1 (0.47) SQORKDM4EHPGDMAPTSMN1; SMN2
SCHEMBL15775763 0.77 SQOR (0.49) SQORADORA2AKDM4EALDH1A1KMT2A
SCHEMBL15775195 0.76 HSP90AA1 (0.47) CYP1A2NR1I3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed