SCHEMBL15775442

SCHEMBL15775442

COc1nc(-c2cccc(C#N)c2)cc2c(N)cccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SQOR Q9Y6N5 7/20 0.48
XDH P47989 1/20 0.47
ADORA2A P29274 2/20 0.44
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
MEN1 O00255 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 2/20 0.42
CLK4 Q9HAZ1 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
PTGDR Q13258 1/20 0.41
BRAF P15056 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775763 0.89 SQOR (0.49) SQORADORA2AMEN1KMT2AALDH1A1
SCHEMBL15775799 0.82 SQOR (0.54) SQORADORA2AMEN1CYP1A2CYP3A4
SCHEMBL15775605 0.81 NR1I3 (0.53) SQOR
SCHEMBL15775231 0.80 SQOR (0.43) SQORXDHCTSSCTSKMEN1
SCHEMBL15775748 0.78 SQOR (0.53) SQORALDH1A1ACP1IDO1
SCHEMBL15775546 0.78 XDH (0.47) SQORXDHCTSSCTSKALDH1A1
SCHEMBL15775389 0.76 ESR1 (0.45) SQORADORA2AMEN1CYP1A2CYP3A4
SCHEMBL15775248 0.73 PARP1 (0.47) SQORACP1IDO1
SCHEMBL15775195 0.72 HSP90AA1 (0.47) CYP1A2CYP2C19CLK4ALDH1A1
SCHEMBL7019095 0.72 ADORA1 (0.60) SQORADORA2AMEN1KMT2ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed