SCHEMBL15775389

SCHEMBL15775389

COc1nc(-c2ccc(O)cc2)cc2c(N)cccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
BLM P54132 1/20 0.42
ALDH1A1 P00352 2/20 0.41
POLB P06746 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SQOR Q9Y6N5 6/20 0.40
KDM4E B2RXH2 1/20 0.40
IDH1 O75874 1/20 0.40
NTSR1 P30989 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
SYK P43405 1/20 0.39
PARP1 P09874 1/20 0.39
TACR3 P29371 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15775748 0.87 SQOR (0.53) ALDH1A1HPGDHSD17B10SQORKDM4E
SCHEMBL15775763 0.83 SQOR (0.49) MEN1KMT2AALDH1A1MAPTSQOR
SCHEMBL15775248 0.83 PARP1 (0.47) MAPTHPGDSQORKDM4EPARP1
SCHEMBL15775799 0.81 SQOR (0.54) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL15775605 0.80 NR1I3 (0.53) SQORTACR3
SCHEMBL15775442 0.76 SQOR (0.48) MEN1KMT2AALDH1A1SQORADORA2A
SCHEMBL15775546 0.76 XDH (0.47) ALDH1A1HPGDHSD17B10SQORKDM4E
SCHEMBL15775195 0.76 HSP90AA1 (0.47) ALDH1A1CYP1A2CYP2C19GSK3AGSK3B
SCHEMBL15775105 0.75 SQOR (0.53) ALDH1A1HPGDHSD17B10SQORKDM4E
SCHEMBL15775484 0.74 L3MBTL1 (0.48) ALDH1A1HPGDHSD17B10SQORTACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014087165-A1 TANKYRASE INHIBITORS UNIVERSITY OF BATH (GB) 2014-06-12 WO disclosed