SCHEMBL15902132

SCHEMBL15902132

CC(C)(C)[Si](C)(C)OCCCc1ccc2[nH]cc(C(=O)Cc3ccc(F)cc3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.39
GABRB2 P47870 3/20 0.39
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
HAT1 O14929 2/20 0.37
EP300 Q09472 2/20 0.37
LMNA P02545 4/20 0.36
RAB9A P51151 3/20 0.36
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
MITF O75030 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HIF1A Q16665 2/20 0.36
XBP1 P17861 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15902481 0.85 GABRA1 (0.45) GABRA1GABRB2HAT1EP300LMNA
SCHEMBL15901066 0.78 HAT1 (0.47) GABRA1GABRB2ALDH1A1SMN1; SMN2HAT1
SCHEMBL15902544 0.77 LMNA (0.42) ALDH1A1HAT1EP300LMNARAB9A
SCHEMBL28604379 0.75 HTR1A (0.34)
SCHEMBL7733863 0.74 MPO (0.56) KMT2A
SCHEMBL2403214 0.73 MAPT (0.46) GABRA1GABRB2MAPTMEN1KMT2A
SCHEMBL15901976 0.72 SLC6A2 (0.35) GABRA1GABRB2ALDH1A1MAPTMEN1
SCHEMBL13894643 0.71 GABRA1 (0.67) GABRA1GABRB2ALDH1A1MEN1KMT2A
SCHEMBL13894640 0.70 KDM4E (0.51) ALDH1A1SMN1; SMN2LMNAMAPTMEN1
SCHEMBL15902273 0.70 GABRA1 (0.55) GABRA1GABRB2ALDH1A1HAT1EP300

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12012411-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2024-06-18 US disclosed
US-20220106321-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-04-07 US disclosed
US-11279704-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-03-22 US disclosed
EP-3617192-A1 VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven K.U. Leuven R&D (BE) 2020-03-04 EP disclosed
US-10550123-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2020-02-04 US disclosed
US-20190337954-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2019-11-07 US disclosed
EP-2760831-B1 VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH (BE) 2019-08-07 EP disclosed
US-20140213586-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2014-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140213586-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885
US-11279704-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885
US-20190337954-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885
US-10550123-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885
US-20220106321-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885
US-12012411-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 GABRA1 4617/4885GABRB2 4748/4885ALDH1A1 4277/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.