SCHEMBL15972715

SCHEMBL15972715

Cc1ccccc1-c1ccc(-c2ccc3nnn(C(N)=O)c3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 4/20 0.43
AMY1A P0DUB6 4/20 0.43
GAA P10253 4/20 0.43
SI P14410 4/20 0.43
MGAM2 Q2M2H8 4/20 0.43
KCNMA1 Q12791 2/20 0.39
TDO2 P48775 1/20 0.39
CTSD P07339 1/20 0.39
BACE1 P56817 1/20 0.39
MGLL Q99685 2/20 0.38
FAAH O00519 1/20 0.38
LCK P06239 1/20 0.38
KDR P35968 1/20 0.38
JAK3 P52333 1/20 0.38
MAPK14 Q16539 1/20 0.38
NMT2 O60551 1/20 0.38
NMT1 P30419 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15973817 0.90 KCNMA1 (0.50) MGAMAMY1AGAASIMGAM2
SCHEMBL15973447 0.89 MGAM (0.47) MGAMAMY1AGAASIMGAM2
SCHEMBL17910001 0.79 SLC9A1 (0.49) TDO2CTSDBACE1LCKKDR
SCHEMBL15973672 0.79 KCNMA1 (0.54) MGAMAMY1AGAASIMGAM2
SCHEMBL443991 0.71 GAA (0.64) MGAMAMY1AGAASIMGAM2
SCHEMBL17909970 0.70 TDO2 (0.54) KCNMA1TDO2CTSDBACE1
SCHEMBL29717601 0.70 MCL1 (0.40) KCNMA1CTSDBACE1MGLLCA12
SCHEMBL15974286 0.70 MCL1 (0.40) BACE1MGLLJAK3CA12CA1
SCHEMBL15973598 0.70 MCL1 (0.40) KCNMA1CTSDBACE1MGLLCA12
SCHEMBL17909968 0.68 CTSD (0.44) CTSDBACE1LCKKDRJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019482-A2 TRISUBSTITUTED BENZOTRIAZOLE DERIVATIVES AS DIHYDROOROTATE OXYGENASE INHIBITORS Aurigene Discovery Technologies Limited (IN) 2016-05-18 EP disclosed
WO-2014128669-A2 TRISUBSTITUTED BENZOTRIAZOLE DERIVATIVES AS DIHYDROOROTATE OXYGENASE INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-08-28 WO disclosed