SCHEMBL1606348

SCHEMBL1606348

COc1ccc2ccccc2c1-c1c(P(c2ccccc2)c2ccccc2)ccc2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.67
KMT2A Q03164 5/20 0.46
MEN1 O00255 4/20 0.46
NISCH Q9Y2I1 1/20 0.46
ALDH1A1 P00352 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NQO1 P15559 1/20 0.43
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29834220 1.00 MAPT (0.67) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL29496547 1.00 MAPT (0.67) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL12446367 0.91 MAPT (0.54) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL7804747 0.89 MAPT (0.59) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL7799304 0.87 MAPT (0.53) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL24779254 0.87 MAPT (0.51) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL4923947 0.87 MAPT (0.65) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL4923948 0.87 MAPT (0.65) MAPTKMT2AMEN1NISCHALDH1A1
SCHEMBL7809875 0.86 MAPT (0.47) MAPTKMT2AMEN1ALDH1A1RAB9A
SCHEMBL146878 0.85 ALDH1A1 (0.44) MAPTALDH1A1KDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 391 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12162829-B2 Gas phase process for acrylate production from ethylene and carbon dioxide CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2024-12-10 US claimed
US-11685755-B2 Dicarbonyl ruthenium and osmium catalysts Universita′ degli Studi di Udine (IT) 2023-06-27 US claimed
US-20230192586-A1 GAS PHASE PROCESS FOR ACRYLATE PRODUCTION FROM ETHYLENE AND CARBON DIOXIDE CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2023-06-22 US claimed
WO-2023114926-A1 GAS PHASE PROCESS FOR ACRYLATE PRODUCTION FROM ETHYLENE AND CARBON DIOXIDE CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2023-06-22 WO claimed
US-11577233-B2 Monocarbonyl ruthenium and osmium catalysts Universita' Delgi Studi Di Udine (IT) 2023-02-14 US claimed
US-11530177-B2 Formation of α,β-unsaturated carboxylic acids and salts thereof from metalalactones and anionic polyelectrolytes CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2022-12-20 US claimed
US-20220168720-A1 MONOCARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIV DEGLI STUDI UDINE (IT) 2022-06-02 US claimed
US-11278876-B2 Monocarbonyl ruthenium and osmium catalysts Universtia Degli Studi Di Udine (IT) 2022-03-22 US claimed
CN-113943318-A Synthesis method of chiral phenyl silanol and 1, 2-chiral disilicon compound 宁夏大学 2022-01-18 CN claimed
CN-113402375-A Formation of alpha, beta-unsaturated carboxylic acids and salts thereof from metallolactones and anionic polyelectrolytes 切弗朗菲利浦化学公司 2021-09-17 CN claimed
EP-3411346-B1 DICARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIV DEGLI STUDI UDINE (IT) 2021-04-28 EP claimed
US-20210107929-A1 DICARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIVERSITA' DEGLI STUDI DI UDINE AND INNOVATION FACTORY S.R.L. (IT) 2021-04-15 US claimed
EP-3411347-B1 MONOCARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIV DEGLI STUDI UDINE (IT) 2021-03-31 EP claimed
US-10941101-B2 Formation of alpha,beta-unsaturated carboxylic acids and salts thereof from metalalactones and anionic polyelectrolytes CHEVRON PHILLIPS CHEMICAL COMPANY, LP (US) 2021-03-09 US claimed
US-20190345089-A1 FORMATION OF ALPHA,BETA-UNSATURATED CARBOXYLIC ACIDS AND SALTS THEREOF FROM METALALACTONES AND ANIONIC POLYELECTROLYTES CHEVRON PHILLIPS CHEMICAL COMPANY LP (US) 2019-11-14 US claimed
US-20190030522-A1 MONOCARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIVERSITA' DEGLI STUDI DI UDINE AND INNOVATION FACTORY S.R.L. (IT) 2019-01-31 US claimed
EP-3411346-A1 DICARBONYL RUTHENIUM AND OSMIUM CATALYSTS Universita' Degli Studi di Udine (IT) 2018-12-12 EP claimed
WO-2017134620-A1 DICARBONYL RUTHENIUM AND OSMIUM CATALYSTS UNIVERSITA' DEGLI STUDI DI UDINE (IT) 2017-08-10 WO claimed
EP-3049072-A1 SYNTHESIS OF DELTA 12-PGJ3 AND RELATED COMPOUNDS William Marsh Rice University (US) 2016-08-03 EP claimed
WO-2015048268-A1 SYNTHESIS OF DELTA 12-PGJ3 AND RELATED COMPOUNDS WILLIAM MARSH RICE UNIVERSITY (US) 2015-04-02 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190345089-A1 FORMATION OF ALPHA,BETA-UNSATURATED CARBOXYLIC ACIDS AND SALTS THEREOF FROM METALALACTONES AND ANIONIC POLYELECTROLYTES ALOX12, ME1, RARA MAPT 2714/4885KMT2A 1907/4885MEN1 4183/4885
US-12162829-B2 Gas phase process for acrylate production from ethylene and carbon dioxide MSMO1, ALOX15, ALOX12 MAPT 1585/4885KMT2A 2885/4885MEN1 612/4885
US-10941101-B2 Formation of alpha,beta-unsaturated carboxylic acids and salts thereof from metalalactones and anionic polyelectrolytes ALOX12, ME1, RARA MAPT 2714/4885KMT2A 1907/4885MEN1 4183/4885
US-11685755-B2 Dicarbonyl ruthenium and osmium catalysts OTC, ODC1, CBR3 MAPT 2422/4885KMT2A 2714/4885MEN1 3163/4885
US-11278876-B2 Monocarbonyl ruthenium and osmium catalysts OTC, CBR3, IDH2 MAPT 2021/4885KMT2A 1600/4885MEN1 1336/4885
US-11530177-B2 Formation of α,β-unsaturated carboxylic acids and salts thereof from metalalactones and anionic polyelectrolytes ME1, ACSL1, ALOX12 MAPT 2510/4885KMT2A 2211/4885MEN1 3606/4885
US-20230192586-A1 GAS PHASE PROCESS FOR ACRYLATE PRODUCTION FROM ETHYLENE AND CARBON DIOXIDE MSMO1, ALOX15, ALOX12 MAPT 1585/4885KMT2A 2885/4885MEN1 612/4885
US-20220168720-A1 MONOCARBONYL RUTHENIUM AND OSMIUM CATALYSTS OTC, CBR3, IDH2 MAPT 2021/4885KMT2A 1600/4885MEN1 1336/4885
US-20210107929-A1 DICARBONYL RUTHENIUM AND OSMIUM CATALYSTS OTC, ODC1, CBR3 MAPT 2422/4885KMT2A 2714/4885MEN1 3163/4885
US-11577233-B2 Monocarbonyl ruthenium and osmium catalysts OTC, CBR3, IDH2 MAPT 2021/4885KMT2A 1600/4885MEN1 1336/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.