SCHEMBL1615

SCHEMBL1615

C[Si](C)(C)CCOC(=O)c1ccccc1-c1ccc(C=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 3/20 0.51
SCN2A Q99250 3/20 0.51
SCN3A Q9NY46 3/20 0.51
SLC6A3 Q01959 3/20 0.42
SLC6A4 P31645 2/20 0.42
ERN1 O75460 1/20 0.41
ALDH1A1 P00352 4/20 0.41
DRD1 P21728 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
DRD3 P35462 1/20 0.41
TSHR P16473 4/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 1/20 0.38
HSP90AA1 P07900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2302 0.85 SCN1A (0.51) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL2127 0.84 SCN1A (0.50) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL3202 0.82 SCN1A (0.51) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL14455157 0.78 ALDH1A1 (0.47) ERN1ALDH1A1TSHRTDP1L3MBTL1
SCHEMBL3293011 0.78 ALDH1A1 (0.54) SCN1ASCN2ASCN3AALDH1A1TSHR
SCHEMBL707956 0.78 SLC6A3 (0.67) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL1614 0.75 SCN1A (0.47) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL17301990 0.75 CA12 (0.43) ALDH1A1TDP1L3MBTL1CYP1A2HSP90AA1
SCHEMBL9569998 0.74 SLC6A3 (0.47) SCN1ASCN2ASCN3ASLC6A3SLC6A4
SCHEMBL25054408 0.73 L3MBTL1 (0.52) ALDH1A1TSHRTDP1L3MBTL1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed