SCHEMBL16158477

SCHEMBL16158477

Cc1ccc(N(c2ccc(C)cc2)c2ccc(N(c3ccc(N(c4ccc(C)cc4)c4ccc(C)cc4)cc3)c3ccc(N(c4ccc(C)cc4)c4cccc(C)c4)cc3)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.48
HSD17B1 P14061 3/20 0.42
HSD17B2 P37059 3/20 0.42
ALDH1A1 P00352 4/20 0.42
TSHR P16473 3/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TP53 P04637 1/20 0.41
GPX4 P36969 1/20 0.41
PAX8 Q06710 1/20 0.41
TDP1 Q9NUW8 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NSD2 O96028 1/20 0.40
CASP3 P42574 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL403133 1.00 ACHE (0.48) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL19075300 1.00 ACHE (0.48) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL3441917 1.00 ACHE (0.48) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL10066016 1.00 ACHE (0.48) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL7741726 0.98 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL11331014 0.96 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL10065418 0.96 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL12957236 0.96 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL13764958 0.96 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR
SCHEMBL2611153 0.96 ACHE (0.46) ACHEHSD17B1HSD17B2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4075533-B1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CANON KK (JP) 2024-07-03 EP disclosed
US-20230320122-A1 ORGANIC LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, IMAGE PICKUP APPARATUS, ELECTRONIC APPARATUS, ILLUMINATION APPARATUS, MOVING OBJECT, AND IMAGE-FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2023-10-05 US disclosed
US-20230320122-A1 ORGANIC LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, IMAGE PICKUP APPARATUS, ELECTRONIC APPARATUS, ILLUMINATION APPARATUS, MOVING OBJECT, AND IMAGE-FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2023-10-05 US disclosed
EP-4255150-A1 ORGANIC LIGHT-EMITTING ELEMENT, LIGHT-EMITTING DEVICE, DISPLAY APPARATUS, IMAGE PICKUP APPARATUS, ELECTRONIC APPARATUS, ILLUMINATION APPARATUS, MOVING OBJECT, AND IMAGE-FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2023-10-04 EP disclosed
US-11672171-B2 Light-emitting device including a plurality of organic electroluminescent elements CANON KABUSHIKI KAISHA (JP) 2023-06-06 US disclosed
US-11672171-B2 Light-emitting device including a plurality of organic electroluminescent elements CANON KABUSHIKI KAISHA (JP) 2023-06-06 US disclosed
EP-2981993-B1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CANON KK (JP) 2022-05-11 EP disclosed
US-20210202848-A1 LIGHT-EMITTING DEVICE INCLUDING A PLURALITY OF ORGANIC ELECTROLUMINESCENT ELEMENTS CANON KK (JP) 2021-07-01 US disclosed
US-10985323-B2 Light-emitting device including a plurality of organic electroluminescent elements CANON KABUSHIKI KAISHA (JP) 2021-04-20 US disclosed
US-20190123279-A1 LIGHT-EMITTING DEVICE INCLUDING A PLURALITY OF ORGANIC ELECTROLUMINESCENT ELEMENTS CANON KABUSHIKI KAISHA (JP) 2019-04-25 US disclosed
US-9911921-B2 Organic compound and organic light-emitting device CANON KABUSHIKI KAISHA (JP) 2018-03-06 US disclosed
US-9911921-B2 Organic compound and organic light-emitting device CANON KABUSHIKI KAISHA (JP) 2018-03-06 US disclosed
US-9755165-B2 Silsesquioxane compound, organic light emitting element, display apparatus, image information processing apparatus, and image forming apparatus CANON KABUSHIKI KAISHA (JP) 2017-09-05 US disclosed
US-9755165-B2 Silsesquioxane compound, organic light emitting element, display apparatus, image information processing apparatus, and image forming apparatus CANON KABUSHIKI KAISHA (JP) 2017-09-05 US disclosed
US-20160118607-A1 SILSESQUIOXANE COMPOUND, ORGANIC LIGHT EMITTING ELEMENT, DISPLAY APPARATUS, IMAGE INFORMATION PROCESSING APPARATUS, AND IMAGE FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-04-28 US disclosed
US-20160118607-A1 SILSESQUIOXANE COMPOUND, ORGANIC LIGHT EMITTING ELEMENT, DISPLAY APPARATUS, IMAGE INFORMATION PROCESSING APPARATUS, AND IMAGE FORMING APPARATUS CANON KABUSHIKI KAISHA (JP) 2016-04-28 US disclosed
US-20150372238-A1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CANON KABUSHIKI KAISHA (JP) 2015-12-24 US disclosed
US-20150372238-A1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CANON KABUSHIKI KAISHA (JP) 2015-12-24 US disclosed
WO-2014163211-A1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE CANON KABUSHIKI KAISHA (JP) 2014-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11672171-B2 Light-emitting device including a plurality of organic electroluminescent elements L1CAM, KCNQ4, SELE ACHE 1779/4885HSD17B1 4636/4885HSD17B2 4397/4885
US-20150372238-A1 ORGANIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE ORC3, AOC3, EML4 ACHE 321/4885HSD17B1 2801/4885HSD17B2 2260/4885
US-20160118607-A1 SILSESQUIOXANE COMPOUND, ORGANIC LIGHT EMITTING ELEMENT, DISPLAY APPARATUS, IMAGE INFORMATION PROCESSING APPARATUS, AND IMAGE FORMING APPARATUS SFXN1, LSS, SLC7A5 ACHE 2810/4885HSD17B1 1667/4885HSD17B2 1370/4885
US-10985323-B2 Light-emitting device including a plurality of organic electroluminescent elements L1CAM, ELOVL6, ELP1 ACHE 1906/4885HSD17B1 4657/4885HSD17B2 4397/4885
US-20210202848-A1 LIGHT-EMITTING DEVICE INCLUDING A PLURALITY OF ORGANIC ELECTROLUMINESCENT ELEMENTS L1CAM, KCNQ4, SELE ACHE 1779/4885HSD17B1 4636/4885HSD17B2 4397/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.