SCHEMBL16182201

SCHEMBL16182201

O=C1CC(c2ccccc2)C2(CCNCC2)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.40
SIGMAR1 Q99720 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.37
OPRM1 P35372 1/20 0.37
SLC18A3 Q16572 1/20 0.37
LMNA P02545 1/20 0.36
DRD2 P14416 1/20 0.36
CTRC Q99895 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
HTR6 P50406 2/20 0.35
KDM1A O60341 3/20 0.35
MAOB P27338 2/20 0.35
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
CA2 P00918 1/20 0.33
OPRK1 P41145 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6006756 0.79 OPRD1 (0.39) OPRD1SIGMAR1HSD17B10OPRM1SLC18A3
SCHEMBL11275319 0.79 CHRM1 (0.43) SIGMAR1SMN1; SMN2DRD2MAPK1KDM1A
SCHEMBL9963267 0.76 CYP2D6 (0.44) SMN1; SMN2MAPK1KDM1AKCNH2
SCHEMBL9644214 0.74 NFKB1 (0.40) SMN1; SMN2HSD17B10CTRCKDM1AMAOB
SCHEMBL12835956 0.74 DRD2 (0.47) SIGMAR1OPRM1DRD2KCNH2
SCHEMBL11282611 0.73 LMNA (0.52) SIGMAR1OPRM1LMNADRD2KCNH2
SCHEMBL11364638 0.72 OPRD1 (0.40) OPRD1SIGMAR1HSD17B10OPRM1SLC18A3
SCHEMBL10748346 0.71 KDM1A (0.46) CTRCALDH1A1KDM1AMAOBNFKB1
SCHEMBL11276382 0.70 BRD4 (0.47) SMN1; SMN2ALDH1A1
SCHEMBL17968386 0.69 SIGMAR1 (0.44) OPRD1SIGMAR1HSD17B10OPRM1SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470021-B1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME (US) 2014-10-22 EP disclosed