SCHEMBL16200051

SCHEMBL16200051

CCn1nc(-c2ccccc2F)c(Cl)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
CNR2 P34972 1/20 0.35
POLB P06746 3/20 0.34
MAPK14 Q16539 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
GAA P10253 1/20 0.33
GNRHR P30968 1/20 0.33
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
MBNL1 Q9NR56 1/20 0.33
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200058 0.81 HSD11B1 (0.40) POLBMAPTTP53KDM4EHPGD
SCHEMBL14044106 0.76 PTGS2 (0.43) PTGS2PTGS1MAPTGAALMNA
SCHEMBL16200214 0.69 ADORA2A (0.40) PTGS2PTGS1RECQLKDM4EALDH1A1
SCHEMBL13066184 0.67 PTGS2 (0.33) PTGS2PTGS1
SCHEMBL16200388 0.67 THRB (0.45) POLBRECQLTDP1MAPTTP53
SCHEMBL16200046 0.67 MEN1 (0.41) PTGS2PTGS1KDM4EALDH1A1HSD11B1
SCHEMBL16200074 0.67 POLB (0.40) PTGS2PTGS1POLBLMNAMBNL1
SCHEMBL16200208 0.67 MAPK1 (0.44) PTGS2PTGS1TDP1MAPTKDM4E
SCHEMBL27894720 0.66 POLB (0.45) POLBRECQLTDP1MAPTLMNA
SCHEMBL8569766 0.66 HSD11B1 (0.47) CNR2MAPK14MAPTNR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed