SCHEMBL16200076

SCHEMBL16200076

Cc1nn(C)c(N2CCNCC2)c1Cl

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
BPTF Q12830 1/20 0.39
NMT1 P30419 6/20 0.37
NMT2 O60551 1/20 0.37
KCNH2 Q12809 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
ADRB2 P07550 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
PDE10A Q9Y233 1/20 0.36
ADRB1 P08588 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16200255 0.83 SMN1; SMN2 (0.38) SMN1; SMN2PDE10AKDM4ECHRM4
SCHEMBL16200075 0.81 LMNA (0.41) NMT1HRH4SMN1; SMN2KDM4E
SCHEMBL16200050 0.71 PDE10A (0.42) CHRNB2CHRNA4BPTFNMT1NMT2
SCHEMBL13184133 0.71 SIGMAR1 (0.39) NMT1SMN1; SMN2KDM4ECHRM2CHRM1
SCHEMBL25146239 0.68 L3MBTL1 (0.46) NMT1SMN1; SMN2KDM4EALDH1A1CHRM2
SCHEMBL14044159 0.68 DRD2 (0.38) SMN1; SMN2KDM4EALDH1A1
SCHEMBL13184164 0.67 ADORA2A (0.36) SMN1; SMN2KDM4EALDH1A1
SCHEMBL14043926 0.67 GABRA1 (0.41) NMT1SMN1; SMN2PDE10AKDM4EALDH1A1
SCHEMBL23964360 0.67 HTR2C (0.50) CHRNB2CHRNA4PDE10AALDH1A1
SCHEMBL25695650 0.66 CYP1A2 (0.48) CHRNB2CHRNA4HRH4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed