Pheniprazine

Pheniprazine

SCHEMBL163709

CC(Cc1ccccc1)NN

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.65
TAAR1 Q96RJ0 5/20 0.65
SLC18A2 Q05940 1/20 0.65
SLC6A2 P23975 2/20 0.58
MAOA P21397 1/20 0.58
SLC6A4 P31645 1/20 0.58
SLC6A3 Q01959 1/20 0.58
CYP2A6 P11509 1/20 0.58
ADORA2A P29274 1/20 0.58
ADORA1 P30542 1/20 0.58
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
CYP2D6 P10635 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
TSHR P16473 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pheniprazine SCHEMBL28842219 1.00 SIGMAR1 (0.65) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
Pheniprazine SCHEMBL13063297 1.00 SIGMAR1 (0.65) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
Pheniprazine SCHEMBL289106 0.98 SIGMAR1 (0.63) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
Pheniprazine SCHEMBL7339052 0.98 SIGMAR1 (0.63) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
Benz(B)Anthracene SCHEMBL11128871 0.89 SIGMAR1 (0.53) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
Pheniprazine SCHEMBL10867258 0.89 NPC1 (0.56) SIGMAR1TAAR1SLC18A2MEN1KMT2A
SCHEMBL30624762 0.81 SIGMAR1 (0.71) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
SCHEMBL21243273 0.81 SIGMAR1 (0.73) SIGMAR1TAAR1SLC18A2SLC6A2MAOA
SCHEMBL8720303 0.80 ACACB (0.47) SIGMAR1TAAR1SLC18A2SLC6A4CYP2A6
Methamphetamine SCHEMBL42615 0.79 SIGMAR1 (1.00) SIGMAR1TAAR1SLC18A2SLC6A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1110 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250339403-A1 Tryptamine Formulations and Uses Thereof Natural MedTech Pty Ltd (AU) 2025-11-06 US claimed
EP-4618981-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE Remedi, Inc. (US) 2025-09-24 EP claimed
EP-4615444-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural Medtech Pty Ltd (AU) 2025-09-17 EP claimed
WO-2025151884-A1 USE OF GLYCOSAMINOGLYCAN SULFATED POLYSACCHARIDES SUCH AS SODIUM PENTOSAN POLYSULFATE IN COMBINATION WITH PERMEATION AGENTS TO TREAT ALZHEIMER'S DISEASE PARSONS C LOWELL (US) 2025-07-17 WO claimed
EP-4479032-A1 NEUROACTIVE STEROIDS FOR TREATMENT OF CNS-RELATED DISORDERS Sage Therapeutics, Inc. (US) 2024-12-25 EP claimed
US-12121513-B2 Betahistine, or a pharmaceutically acceptable salt thereof, and a monoamine oxidase inhibitor, for use in the treatment or prevention of one or more symptoms of vertigo in a subject Intrabio Ltd. (GB) 2024-10-22 US claimed
WO-2024108195-A1 COMBINATIONS OF MONOAMINE OXIDASE INHIBITORS AND SEROTONIN RECEPTOR AGONISTS AND THEIR THERAPEUTIC USE REMEDI, INC. (US) 2024-05-23 WO claimed
WO-2024098098-A1 TRYPTAMINE FORMULATIONS AND USES THEREOF Natural MedTech Pty Ltd (AU) 2024-05-16 WO claimed
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION ANEUROTECH BV (BE) 2023-11-30 US claimed
US-20230364115-A1 NOVEL PSYCHEDELIC COMPOSITIONS, DELIVERY SYSTEMS AND THERAPEUTIC USES THEREOF MYDECINE INNOVATIONS GROUP INC (US) 2023-11-16 US claimed
EP-0797442-B1 TREATMENT OF OPTIC NEURITIS MASSACHUSETTS EYE & EAR INFIRM (US) 2003-05-21 EP claimed
US-20020161016-A1 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation VIVUS LLC (F/K/A VIVUS, INC.) 2002-10-31 US claimed
WO-2002041883-A2 AS-NEEDED ADMINISTRATION OF TRICYCLIC AND OTHER NON-SRI ANTIDEPRESSANT DRUGS TO TREAT PREMATURE EJACULATION VIVUS, INC. (US) 2002-05-30 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0070832-A4 MICROENCAPSULATED FLUORESCER COMPOSITION, TEST KIT AND SYSTEM FOR IMMUNOASSAY. ELECTRO NUCLEONICS (US) 1983-06-17 EP claimed
EP-0070832-A1 MICROENCAPSULATED FLUORESCER COMPOSITION, TEST KIT AND SYSTEM FOR IMMUNOASSAY ELECTRO-NUCLEONICS, INC. (US) 1983-02-09 EP claimed
US-4372745-A QUALITATIVE AND QUANTITATIVE ANALYSIS ELECTRO-NUCLEONICS, INC. (US) 1983-02-08 US claimed
WO-1982002772-A1 MICROENCAPSULATED FLUORESCER COMPOSITION,TEST KIT AND SYSTEM FOR IMMUNOASSAY ELECTRO NUCLEONICS (US) 1982-08-19 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020161016-A1 As-needed administration of tricyclic and other non-SRI antidepressant drugs to treat premature ejaculation HTR5A, HTR1A, MAOA SIGMAR1 11/4885TAAR1 150/4885SLC18A2 35/4885
US-20230381168-A1 ADJUNCTIVE THERAPY FOR DEPRESSION HTR2A, HTR3B, HTR5A SIGMAR1 174/4885TAAR1 49/4885SLC18A2 46/4885
US-12121513-B2 Betahistine, or a pharmaceutically acceptable salt thereof, and a monoamine oxidase inhibitor, for use in the treatment or prevention of one or more symptoms of vertigo in a subject HNMT, MAOA, MAOB SIGMAR1 1620/4885TAAR1 655/4885SLC18A2 30/4885
US-20250339403-A1 Tryptamine Formulations and Uses Thereof MAOA, MAOB, TPH1 SIGMAR1 563/4885TAAR1 55/4885SLC18A2 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.