SCHEMBL16503545

SCHEMBL16503545

CC=C(OC)c1ccc2cccc(-c3cccc4cccnc34)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.40
CCR1 P32246 3/20 0.40
CCR5 P51681 3/20 0.40
CCR8 P51685 3/20 0.40
HTT P42858 3/20 0.40
MAPT P10636 2/20 0.40
MMP9 P14780 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP3A4 P08684 2/20 0.40
ALOX15 P16050 2/20 0.40
GMNN O75496 1/20 0.40
TP53 P04637 1/20 0.40
HSP90AA1 P07900 1/20 0.40
MMP2 P08253 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
MMP8 P22894 1/20 0.40
THPO P40225 1/20 0.40
MTOR P42345 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16502605 0.84 ALOX15 (0.56) LMNAHTTMAPTKDM4EALOX15
SCHEMBL7920176 0.78 CCR1 (0.46) LMNACCR1CCR5CCR8HTT
SCHEMBL16502608 0.78 SLC40A1 (0.50) LMNACCR1CCR5CCR8HTT
SCHEMBL7919762 0.76 KDM4E (0.34) LMNAMAPTKDM4ESMN1; SMN2MEN1
SCHEMBL16503574 0.74 GABRG2 (0.33) MAPTKDM4ETP53HSP90AA1SMN1; SMN2
SCHEMBL7916651 0.72 TUBB4A (0.38) KDM4EMEN1KMT2AHDAC8HDAC6
SCHEMBL16502784 0.72 SLC9A1 (0.48)
SCHEMBL16502512 0.70 ALOX15 (0.54) HTTMAPTKDM4EALOX15TP53
SCHEMBL7916645 0.70 HDAC6 (0.42) LMNAHTTMAPTALOX15HDAC3
SCHEMBL16502596 0.70 ALOX15 (0.61) HTTMAPTKDM4EALOX15TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394987-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2011-12-14 EP disclosed