SCHEMBL16600110

SCHEMBL16600110

NC(=O)c1ccc(-c2cccc(F)c2F)c(N2CCNCC2)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.42
ACVR1 Q04771 1/20 0.41
PARP1 P09874 5/20 0.37
CAMK1D Q8IU85 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
HTR1A P08908 2/20 0.36
HTR7 P34969 1/20 0.36
HTR2B P41595 1/20 0.36
HTR3A P46098 1/20 0.36
HTR6 P50406 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
JAK2 O60674 1/20 0.35
HPGD P15428 1/20 0.35
PRKD3 O94806 1/20 0.35
MAPK9 P45984 1/20 0.35
MAPKAPK2 P49137 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16599760 0.85 ADRB1 (0.43) BTKACVR1MAPK10
SCHEMBL30798658 0.82 ACVR1 (0.45) ACVR1PARP1ALDH1A1LMNA
SCHEMBL25366356 0.72 HTR6 (0.44) ACVR1HTR7HTR6
SCHEMBL3883327 0.71 SMARCA2 (0.42) ACVR1HTR1AHTR7HTR6ALDH1A1
SCHEMBL30311470 0.70 ALB (0.47) HRH4HTR3AALDH1A1LMNAHPGD
SCHEMBL6262440 0.70 RXFP1 (0.42) BTKACVR1HTR7MAPKAPK2MAPK14
SCHEMBL15059858 0.69 NPC1 (0.55) PARP1ALDH1A1JAK2HPGD
SCHEMBL18641223 0.68 PRKCA (0.46) ACVR1PARP1HTR7SLC6A4ALDH1A1
SCHEMBL746343 0.68 ALDH1A1 (0.54) HTR1AHTR7HTR2BHTR3AHTR6
SCHEMBL3633976 0.68 ACVR1 (0.62) ACVR1PARP1HTR1AHTR7HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015048306-A1 NOVEL AGENTS TARGETING CYP51 THE SCRIPPS RESEARCH INSTITUTE (US) 2015-04-02 WO disclosed