SCHEMBL1661047

SCHEMBL1661047

CCC(=O)C1Oc2ccc(CCC(C)C)cc2O1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
PTGS2 P35354 8/20 0.35
PTGS1 P23219 3/20 0.35
HPGD P15428 1/20 0.34
IKBKE Q14164 1/20 0.33
TBK1 Q9UHD2 1/20 0.33
ADRB2 P07550 3/20 0.33
ADRB1 P08588 3/20 0.33
ADRB3 P13945 3/20 0.33
ADRA1D P25100 3/20 0.33
ADRA1A P35348 3/20 0.33
ADRA1B P35368 3/20 0.33
ACACB O00763 2/20 0.32
CACNA1H O95180 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663353 0.86 PTGS2 (0.38) GRIN2DGRIN2AGRIN2BGRIN2CPTGS2
SCHEMBL1661045 0.74 PTGS2 (0.39) PTGS2
SCHEMBL29852250 0.72 PTGS2 (0.40) PTGS2PTGS1HPGD
SCHEMBL1291782 0.72 PTGS2 (0.40) PTGS2PTGS1HPGD
SCHEMBL1292040 0.70 ALDH1A1 (0.46) PTGS2HPGD
SCHEMBL1292093 0.69 ALDH1A1 (0.47) HPGD
SCHEMBL8294114 0.66 TAAR1 (0.61) HPGD
SCHEMBL16978376 0.66 TAAR1 (0.41) PTGS2
SCHEMBL21377531 0.65 ALOX15 (0.54) GRIN2DGRIN2AGRIN2BGRIN2CPTGS2
SCHEMBL15558442 0.65 ALOX15 (0.68) GRIN2DGRIN2AGRIN2BGRIN2CHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2624811-B1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH & CIE (CH) 2017-06-21 EP disclosed
EP-2624811-B1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH & CIE (CH) 2017-06-21 EP disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-8987188-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2015-03-24 US disclosed
US-8987188-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2015-03-24 US disclosed
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2013-10-31 US disclosed
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2013-10-31 US disclosed
WO-2012045646-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2012-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS TRPA1, BBOX1, PAOX GRIN2D 1555/4885GRIN2A 3105/4885GRIN2B 2655/4885
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS BBOX1, CBR3, CBR1 GRIN2D 2092/4885GRIN2A 3606/4885GRIN2B 3018/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.