SCHEMBL1663353

SCHEMBL1663353

CC(=O)C1Oc2ccc(CCC(C)C)cc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.38
GRIN2D O15399 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
PTGS1 P23219 2/20 0.36
ACACB O00763 1/20 0.35
IKBKE Q14164 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
POLB P06746 1/20 0.33
CACNA1H O95180 1/20 0.33
CYP3A4 P08684 1/20 0.33
HPGD P15428 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
ADRB3 P13945 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661047 0.86 GRIN2D (0.35) PTGS2GRIN2DGRIN2AGRIN2BGRIN2C
SCHEMBL29852250 0.83 PTGS2 (0.40) PTGS2PTGS1POLBCYP3A4HPGD
SCHEMBL1291782 0.83 PTGS2 (0.40) PTGS2PTGS1POLBCYP3A4HPGD
SCHEMBL1292040 0.81 ALDH1A1 (0.46) PTGS2POLBHPGD
SCHEMBL1292044 0.75 PTGS2 (0.38) PTGS2POLBCYP3A4HPGD
SCHEMBL1292020 0.75 CYP3A4 (0.47) PTGS2PTGS1POLBCYP3A4HPGD
SCHEMBL1292011 0.72 MCHR1 (0.36) POLBCYP3A4
SCHEMBL1663351 0.72 ALDH1A1 (0.41) PTGS2PTGS1HPGD
SCHEMBL19005894 0.70 PTGS2 (0.35) PTGS2PTGS1POLBCYP3A4
SCHEMBL1291722 0.70 PTGS2 (0.35) PTGS2PTGS1POLBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2624811-B1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH & CIE (CH) 2017-06-21 EP disclosed
EP-2624811-B1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH & CIE (CH) 2017-06-21 EP disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-9382500-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2016-07-05 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2015-06-04 US disclosed
US-8987188-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2015-03-24 US disclosed
US-8987188-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2015-03-24 US disclosed
US-8987188-B2 Benzodioxole derivatives as watery odorants FIRMENICH SA (CH) 2015-03-24 US disclosed
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2013-10-31 US disclosed
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2013-10-31 US disclosed
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2013-10-31 US disclosed
WO-2012045646-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS FIRMENICH SA (CH) 2012-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150152352-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS TRPA1, BBOX1, PAOX PTGS2 771/4885GRIN2D 1555/4885GRIN2A 3105/4885
US-20130288947-A1 BENZODIOXOLE DERIVATIVES AS WATERY ODORANTS BBOX1, CBR3, CBR1 PTGS2 914/4885GRIN2D 2092/4885GRIN2A 3606/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.