SCHEMBL16612656

SCHEMBL16612656

COc1cc2c(ccn2CCn2c[c]c(C(N)=O)n2)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 9/20 0.42
CXCR3 P49682 1/20 0.37
KMO O15229 1/20 0.36
MTNR1A P48039 2/20 0.35
MTNR1B P49286 2/20 0.35
HCRTR1 O43613 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
PHGDH O43175 1/20 0.34
TRPM5 Q9NZQ8 1/20 0.33
HTR4 Q13639 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612831 0.92 HCRTR2 (0.42) HCRTR2MTNR1AMTNR1BHCRTR1TSHR
SCHEMBL16612745 0.88 HDAC6 (0.42) HCRTR2CXCR3KMOHDAC6HDAC1
SCHEMBL16612868 0.83 MTNR1A (0.49) HCRTR2MTNR1AMTNR1BHCRTR1HDAC6
SCHEMBL16612854 0.82 MTNR1A (0.52) HCRTR2MTNR1AMTNR1BHCRTR1HTT
SCHEMBL12480072 0.81 HTR2A (0.41) HCRTR2KMOHDAC6HDAC1HDAC8
SCHEMBL16612628 0.81 HCRTR2 (0.43) HCRTR2MTNR1AMTNR1BHCRTR1
SCHEMBL16612982 0.81 HCRTR2 (0.44) HCRTR2MTNR1AMTNR1BHCRTR1
SCHEMBL16613000 0.79 HTR2A (0.42) HCRTR2MTNR1AMTNR1BHCRTR1HDAC6
SCHEMBL16612997 0.79 HCRTR2 (0.42) HCRTR2MTNR1AMTNR1BHCRTR1TSHR
SCHEMBL16612936 0.77 MTNR1A (0.50) HCRTR2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed