SCHEMBL16612704

SCHEMBL16612704

NC(=O)c1[c]cn(CCn2ccc3ncccc32)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 6/20 0.41
HCRTR2 O43614 1/20 0.37
P2RX7 Q99572 1/20 0.36
RPS6KA5 O75582 1/20 0.34
LMNA P02545 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
PDE4D Q08499 1/20 0.33
EGLN3 Q9H6Z9 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CDC7 O00311 1/20 0.32
CDK2 P24941 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
NR3C1 P04150 1/20 0.31
NR3C2 P08235 1/20 0.31
PSMB5 P28074 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612739 0.83 TDP1 (0.54) LMNAEGLN3TDP1KDM4ENPC1
SCHEMBL16612954 0.82 LMNA (0.53) LMNA
SCHEMBL16612613 0.81 MTNR1A (0.49) HCRTR2P2RX7LMNASLC22A12
SCHEMBL16612920 0.75 CDK4 (0.52) LMNA
SCHEMBL16612745 0.74 HDAC6 (0.42) HCRTR2LMNA
SCHEMBL12480072 0.74 HTR2A (0.41) HCRTR2LMNA
SCHEMBL16612876 0.74 HTR2C (0.41) HCRTR2P2RX7LMNA
SCHEMBL16613000 0.74 HTR2A (0.42) HCRTR2LMNAJAK2JAK1TYK2
SCHEMBL16612960 0.73 HCRTR2 (0.41) METHCRTR2KDM4E
SCHEMBL16612831 0.72 HCRTR2 (0.42) HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed