SCHEMBL16612613

SCHEMBL16612613

NC(=O)c1[c]cn(CCn2ccc3cccnc32)n1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.49
PARP1 P09874 2/20 0.45
DAO P14920 1/20 0.44
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
P2RX7 Q99572 1/20 0.36
SLC22A12 Q96S37 8/20 0.36
LMNA P02545 1/20 0.33
SLC22A6 Q4U2R8 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
ENPP1 P22413 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612954 0.82 LMNA (0.53) MTNR1ADAOLMNA
SCHEMBL16612871 0.81 HCRTR2 (0.36) MTNR1AHCRTR2
SCHEMBL16612704 0.81 MET (0.41) HCRTR2P2RX7SLC22A12LMNA
SCHEMBL16612773 0.79 MTNR1A (0.53) MTNR1APARP1HCRTR1HCRTR2
SCHEMBL16612705 0.78 HCRTR2 (0.38) HCRTR2LMNA
SCHEMBL16612790 0.78 HCRTR2 (0.39) HCRTR2P2RX7LMNA
SCHEMBL16612960 0.77 HCRTR2 (0.41) HCRTR2
SCHEMBL16612920 0.75 CDK4 (0.52) MTNR1ALMNA
SCHEMBL16612745 0.74 HDAC6 (0.42) HCRTR2LMNA
SCHEMBL12480072 0.74 HTR2A (0.41) HCRTR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed