SCHEMBL16612790

SCHEMBL16612790

Cc1cccc2ccn(CCn3c[c]c(C(N)=O)n3)c12

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 2/20 0.39
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
P2RX7 Q99572 1/20 0.36
LMNA P02545 1/20 0.33
CXCR3 P49682 1/20 0.33
PLA2G10 O15496 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HTR1A P08908 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612705 0.86 HCRTR2 (0.38) HCRTR2LMNACXCR3HTR1ASLC6A4
SCHEMBL16612954 0.81 LMNA (0.53) LMNAMAPTSMN1; SMN2
SCHEMBL16613000 0.80 HTR2A (0.42) HCRTR2LMNAMAPT
SCHEMBL16612613 0.78 MTNR1A (0.49) HCRTR2P2RX7LMNA
SCHEMBL16612920 0.74 CDK4 (0.52) LMNASMN1; SMN2
SCHEMBL16612745 0.74 HDAC6 (0.42) HCRTR2LMNACXCR3
SCHEMBL16612871 0.74 HCRTR2 (0.36) HCRTR2CXCR3
SCHEMBL16612831 0.73 HCRTR2 (0.42) HCRTR2
SCHEMBL16612773 0.73 MTNR1A (0.53) HCRTR2CXCR3
SCHEMBL16612868 0.73 MTNR1A (0.49) HCRTR2LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed