SCHEMBL16612705

SCHEMBL16612705

NC(=O)c1[c]cn(CCn2ccc3cccc(F)c32)n1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.38
HTR1A P08908 3/20 0.37
SLC6A4 P31645 2/20 0.37
LMNA P02545 1/20 0.33
CXCR3 P49682 1/20 0.33
CA5A P35218 1/20 0.32
AR P10275 1/20 0.32
FABP4 P15090 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612790 0.86 HCRTR2 (0.39) HCRTR2HTR1ASLC6A4LMNACXCR3
SCHEMBL16612954 0.81 LMNA (0.53) LMNA
SCHEMBL16612613 0.78 MTNR1A (0.49) HCRTR2LMNA
SCHEMBL16612876 0.77 HTR2C (0.41) HCRTR2HTR1ASLC6A4LMNAAR
SCHEMBL16613000 0.75 HTR2A (0.42) HCRTR2LMNAFABP4
SCHEMBL16612920 0.74 CDK4 (0.52) LMNA
SCHEMBL16612871 0.74 HCRTR2 (0.36) HCRTR2CXCR3
SCHEMBL16612745 0.74 HDAC6 (0.42) HCRTR2LMNACXCR3
SCHEMBL12480072 0.73 HTR2A (0.41) HCRTR2LMNA
SCHEMBL16612704 0.71 MET (0.41) HCRTR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed