SCHEMBL1662282

SCHEMBL1662282

CC(C)(C)[Si](C)(C)Oc1cccc(C2CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.46
DRD2 P14416 2/20 0.40
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA9 Q16790 4/20 0.40
ADRA1A P35348 5/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
HTR1A P08908 3/20 0.38
ADRA1D P25100 3/20 0.38
ADRA1B P35368 3/20 0.38
NOTUM Q6P988 1/20 0.35
PREP P48147 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23923489 0.81 HTR2A (0.42) HTR2CCA12CA1CA9HSP90AA1
SCHEMBL23923488 0.81 HTR2A (0.42) HTR2CCA12CA1CA9HSP90AA1
SCHEMBL7706827 0.80 CA1 (0.50) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL3093088 0.78 HSP90AA1 (0.38) HTR2CCA12CA1CA9HSP90AA1
SCHEMBL9988239 0.77 SLC6A4 (0.41) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL3182564 0.75 CA12 (0.46) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL5508174 0.75 CA12 (0.33) HTR2CCA12CA1CA9ADRA1A
SCHEMBL2329760 0.74 ACHE (0.50) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL4004898 0.74 CYP3A4 (0.47) CA12CA1CA9HSP90AA1HSP90AB1
SCHEMBL5292779 0.74 ACHE (0.45) CA12CA1CA9NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12435040-B2 1,3-substituted cyclobutyl derivatives and uses thereof BAUSCH + LOMB IRELAND LIMITED (IE) 2025-10-07 US disclosed
CN-115916763-B Antiviral 1, 3-dioxoindene compounds 诺华股份有限公司 2025-06-03 CN disclosed
US-20250090491-A1 ANTIVIRAL 1,3-DI-OXO-INDENE COMPOUNDS NOVARTIS AG (CH) 2025-03-20 US disclosed
US-20240308965-A1 1,3-SUBSTITUTED CYCLOBUTYL DERIVATIVES AND USES THEREOF JPMORGAN CHASE BANK, N.A., AS SUCCESSOR AGENT 2024-09-19 US disclosed
US-12083092-B2 Antiviral 1,3-di-oxo-indene compounds NOVARTIS AG (CH) 2024-09-10 US disclosed
EP-4313951-A1 1,3-SUBSTITUTED CYCLOBUTYL DERIVATIVES AND USES THEREOF Novartis AG (CH) 2024-02-07 EP disclosed
US-11845730-B2 1,3-substituted cyclobutyl derivatives and uses thereof CITIBANK, N.A., AS NOTES COLLATERAL AGENT 2023-12-19 US disclosed
US-20230382931-A1 DIOXOLANE ANALOGUES OF URIDINE FOR THE TREATMENT OF CANCER MEDIVIR AB (SE) 2023-11-30 US disclosed
CN-117062804-A 1, 3-substituted cyclobutyl derivatives and their use 诺华股份有限公司 2023-11-14 CN disclosed
CN-110790789-B Dioxolane analogues of uridine for use in the treatment of cancer 美迪维尔公司 2023-05-12 CN disclosed
EP-3041855-A1 HCV POLYMERASE INHIBITORS MEDIVIR AB (SE) 2016-07-13 EP disclosed
WO-2016030335-A1 DIOXOLANE ANALOGUES OF URIDINE FOR THE TREATMENT OF CANCER MEDIVIR AB (SE) 2016-03-03 WO disclosed
US-20150175648-A1 HCV POLYMERASE INHIBITORS MEDIVIR AB (SE) 2015-06-25 US disclosed
WO-2015056213-A1 HCV POLYMERASE INHIBITORS MEDIVIR AB (SE) 2015-04-23 WO disclosed
WO-2015034420-A1 HCV POLYMERASE INHIBITORS MEDIVIR AB (SE) 2015-03-12 WO disclosed
EP-2307394-B1 SULPHONAMIDES AS VANILLOID RECEPTOR ANTAGONIST AMOREPACIFIC CORP (KR) 2012-09-26 EP disclosed
US-20110152318-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2011-06-23 US disclosed
US-20110152318-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2011-06-23 US disclosed
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed
WO-2010002209-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2010-01-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11845730-B2 1,3-substituted cyclobutyl derivatives and uses thereof TRPV1, TRPV3, TRPV2 HTR2C 437/4885DRD2 1908/4885CA12 2835/4885
US-12435040-B2 1,3-substituted cyclobutyl derivatives and uses thereof TRPV1, TRPV3, TRPV2 HTR2C 437/4885DRD2 1908/4885CA12 2835/4885
US-20110152318-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME TRPV1, TRPA1, TRPV2 HTR2C 274/4885DRD2 438/4885CA12 3088/4885
US-20240308965-A1 1,3-SUBSTITUTED CYCLOBUTYL DERIVATIVES AND USES THEREOF TRPV1, TRPV3, TRPV2 HTR2C 437/4885DRD2 1908/4885CA12 2835/4885
US-20250090491-A1 ANTIVIRAL 1,3-DI-OXO-INDENE COMPOUNDS IRF3, EIF2AK2, MAVS HTR2C 3176/4885DRD2 4053/4885CA12 3710/4885
US-20150175648-A1 HCV POLYMERASE INHIBITORS POLI, POLB, POLL HTR2C 3877/4885DRD2 2060/4885CA12 4101/4885
US-20230382931-A1 DIOXOLANE ANALOGUES OF URIDINE FOR THE TREATMENT OF CANCER ADORA3, DUT, NTPCR HTR2C 958/4885DRD2 268/4885CA12 3689/4885
US-12083092-B2 Antiviral 1,3-di-oxo-indene compounds IRF3, EIF2AK2, MAVS HTR2C 3176/4885DRD2 4053/4885CA12 3710/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.