SCHEMBL16656240

SCHEMBL16656240

C[Si](C)(C)C#Cc1ccc(N(c2ccc(CO)cc2)c2ccc(CO)cc2)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
ACACB O00763 1/20 0.32
FFAR1 O14842 2/20 0.32
EGLN1 Q9GZT9 1/20 0.32
APP P05067 2/20 0.31
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRA4 P48169 1/20 0.31
GABRA6 Q16445 1/20 0.31
ADK P55263 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1710488 0.89 NOS3 (0.38) NOS3NOS1FFAR1EGLN1GABRA1
SCHEMBL6851297 0.86 GABRA1 (0.33) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL14882956 0.79 ALDH1A1 (0.42) APPGABRA1GABRG2GABRB3GABRA5
SCHEMBL4107898 0.77 APP (0.41) APPGABRA1GABRG2GABRB3GABRA5
SCHEMBL17934728 0.77 ADK (0.37) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL20716885 0.77 NOS3 (0.35) NOS3NOS1FFAR1EGLN1
SCHEMBL3254459 0.76 CYP2A6 (0.50) ACACBFFAR1EGLN1GABRA1GABRG2
SCHEMBL22146946 0.76 NOS3 (0.34) NOS3NOS1FFAR1EGLN1
SCHEMBL308282 0.75 TSHR (0.48) NOS3NOS1MEN1KMT2A
SCHEMBL3345157 0.75 ACACB (0.45) ACACBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9012773-B2 Thiazole-based compound and uses thereof NEC CORPORATION (JP) 2015-04-21 US disclosed