SCHEMBL1669451

SCHEMBL1669451

COC(=O)Cc1ccc(O)c(C2(c3ccccc3)CCNCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
GFER P55789 1/20 0.47
PDK2 Q15119 1/20 0.44
OPRM1 P35372 4/20 0.43
TACR1 P25103 2/20 0.41
TSHR P16473 3/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 1/20 0.39
NFKB1 P19838 2/20 0.39
NPC1 O15118 1/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTR2A P28223 1/20 0.38
HSP90AB1 P08238 1/20 0.38
SLC7A5 Q01650 1/20 0.38
ERCC1 P07992 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12800747 0.89 ALDH1A1 (0.48) ALDH1A1GAAGFERPDK2TACR1
SCHEMBL1669606 0.80 CA12 (0.47) ALDH1A1PDK2OPRM1TSHRHPGD
SCHEMBL1669154 0.79 OPRD1 (0.51) ALDH1A1GAAGFERPDK2TACR1
SCHEMBL12800418 0.76 OPRM1 (0.40) OPRM1TACR1HTR2APTGDR2
SCHEMBL1668446 0.76 OPRM1 (0.47) ALDH1A1GAAOPRM1TACR1TSHR
SCHEMBL24944048 0.74 GAA (0.51) ALDH1A1GAATSHRNFKB1TDP1
SCHEMBL16499058 0.74 KDM1A (0.40) ALDH1A1GAAGFEROPRM1
SCHEMBL24943646 0.74 ERCC1 (0.44) GAAOPRM1TACR1TSHRHPGD
SCHEMBL24943732 0.72 GAA (0.51) ALDH1A1GAAOPRM1TSHRHPGD
SCHEMBL24944632 0.71 CA2 (0.47) OPRM1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed