SCHEMBL16702991

SCHEMBL16702991

CC(C)[CH]OC(=O)Oc1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.43
CYP11B1 P15538 3/20 0.42
CYP11B2 P19099 3/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
ENPP2 Q13822 1/20 0.39
AKR1C3 P42330 3/20 0.39
ELANE P08246 1/20 0.38
MMP2 P08253 2/20 0.38
MMP9 P14780 2/20 0.38
MMP14 P50281 2/20 0.38
AKR1C2 P52895 2/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4196181 0.78 ALDH1A1 (0.41) MAPTELANEKMT2A
SCHEMBL16702992 0.75 CA2 (0.50) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL16703079 0.74 PTGS2 (0.48) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL2294329 0.73 PTGS2 (0.44) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL2294327 0.73 PTGS2 (0.44) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL3234259 0.73 MMP2 (0.42) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL9352386 0.72 ELANE (0.62) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL1930857 0.72 MAPT (0.74) PTGS2POLBMAPTPKMENPP2
SCHEMBL14596348 0.71 THRB (0.53) PTGS2CYP11B1CYP11B2POLBMAPT
SCHEMBL27825837 0.71 PTGS2 (0.50) PTGS2CYP11B1CYP11B2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3066091-A1 NMDA ANTAGONIST PRODRUGS Astrazeneca AB (SE) 2016-09-14 EP disclosed
WO-2015067923-A1 NMDA ANTAGONIST PRODRUGS ASTRAZENECA AB (SE) 2015-05-14 WO disclosed