SCHEMBL16720155

SCHEMBL16720155

Oc1ccc[c]c1-c1cccc(F)c1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.33
BCHE P06276 1/20 0.33
CES1 P23141 1/20 0.33
CNR2 P34972 1/20 0.33
HSD17B14 Q9BPX1 2/20 0.32
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
CA12 O43570 1/20 0.31
GMNN O75496 1/20 0.31
ALDH1A1 P00352 1/20 0.31
EGFR P00533 1/20 0.31
CA2 P00918 1/20 0.31
LMNA P02545 1/20 0.31
FYN P06241 1/20 0.31
POLB P06746 1/20 0.31
CA3 P07451 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
MMP9 P14780 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720271 0.85 MAPT (0.39) KDM4ENPC1CA12GMNNALDH1A1
SCHEMBL12815748 0.83 CCNE2 (0.35) CES2BCHECES1PIK3CASLC9A1
SCHEMBL16720251 0.79 CA2 (0.35) CES2CES1KDM4ENPC1CA12
SCHEMBL2053579 0.79 ACHE (0.39) NPC1RAB9ASMN1; SMN2BCAT1CCNE2
SCHEMBL2014554 0.79 TAAR1 (0.34) KDM4ETDP1BCAT1CCNE2CCNE1
SCHEMBL2373478 0.77 SMN1; SMN2 (0.46) KDM4ENPC1CA12GMNNALDH1A1
SCHEMBL2049471 0.76 HSD11B1 (0.46) CES1
SCHEMBL16720359 0.74 ALDH1A1 (0.40) CES2CES1KDM4EALDH1A1CA2
SCHEMBL6367917 0.72 ALDH1A1 (0.44) CES2BCHECES1HSD17B14KDM4E
SCHEMBL27341090 0.72 MAOA (0.46) CES2BCHECES1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed