SCHEMBL16740674

SCHEMBL16740674

C=CC(=O)C(C)(C)Cc1ccc(Br)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 2/20 0.47
THRB P10828 2/20 0.47
THRA P10827 1/20 0.47
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
LMNA P02545 2/20 0.40
F13A1 P00488 1/20 0.40
TGM1 P22735 1/20 0.40
TGM3 Q08188 1/20 0.40
LSS P48449 2/20 0.38
PYCR1 P32322 1/20 0.38
MME P08473 2/20 0.37
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
EPHX1 P07099 1/20 0.35
BLM P54132 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3136867 0.91 THRB (0.55) TGM2THRBTHRACYP2C19ALDH1A1
SCHEMBL8161806 0.83 THRA (0.47) THRBTHRACYP2C19ALDH1A1CYP3A4
SCHEMBL16740573 0.83 THRA (0.47) TGM2THRBTHRACYP2C19ALDH1A1
SCHEMBL11092024 0.82 CYP3A4 (0.58) THRBTHRACYP2C19ALDH1A1CYP3A4
SCHEMBL9422511 0.81 THRB (0.54) THRBTHRACYP2C19ALDH1A1CYP3A4
SCHEMBL16740537 0.80 ALDH1A1 (0.47) TGM2THRBTHRAALDH1A1CYP3A4
SCHEMBL5149405 0.78 BLM (0.46) ALDH1A1CYP3A4LMNAMMEMEN1
SCHEMBL10767808 0.78 LMNA (0.42) TGM2THRBTHRACYP2C19ALDH1A1
SCHEMBL16740667 0.78 TGM2 (0.45) TGM2THRBTHRACYP2C19ALDH1A1
SCHEMBL3664414 0.76 HTT (0.38) THRBTHRACYP2C19CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015075051-A1 ALLOSTERIC INHIBITORS OF ATYPICAL PROTEIN KINASES C UNIVERSITAET DES SAARLANDES (DE) 2015-05-28 WO disclosed