SCHEMBL1684375

SCHEMBL1684375

O=C1NS(=O)(=O)c2ccc(Br)cc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.62
DAPK3 O43293 1/20 0.62
MAP4K4 O95819 1/20 0.62
RET P07949 1/20 0.62
PIM1 P11309 1/20 0.62
LTK P29376 1/20 0.62
GRK5 P34947 1/20 0.62
CSNK1A1 P48729 1/20 0.62
CDK8 P49336 1/20 0.62
PRKX P51817 1/20 0.62
LIMK1 P53667 1/20 0.62
CDK5 Q00535 1/20 0.62
ACVR1 Q04771 1/20 0.62
PTK2 Q05397 1/20 0.62
TYRO3 Q06418 1/20 0.62
PRKAA1 Q13131 1/20 0.62
DYRK1A Q13627 1/20 0.62
NTRK3 Q16288 1/20 0.62
LRRK2 Q5S007 1/20 0.62
CLK4 Q9HAZ1 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016818 1.00 CHEK1 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL30834838 0.85 CA12 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL1476316 0.85 CA12 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL32689426 0.77 CHEK1 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL29441946 0.77 CHEK1 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL30873095 0.77 CA12 (0.73) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL2208975 0.77 CHEK1 (0.62) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL3988311 0.77 CA12 (0.73) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL3984666 0.77 RET (1.00) CHEK1DAPK3MAP4K4RETPIM1
SCHEMBL1666180 0.77 CHEK1 (0.62) CHEK1DAPK3MAP4K4RETPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026103694-A1 HDAC INHIBITOR, AND PREPARATION AND USE THEREOF 赛岚(杭州)生物医药科技有限公司 2026-05-21 WO disclosed
US-20260092053-A1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2026-04-02 US disclosed
EP-4681774-A2 KHK INHIBITORS Gilead Sciences, Inc. (US) 2026-01-21 EP disclosed
EP-4313967-B1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2025-11-12 EP disclosed
EP-4387965-A2 ARYL SULFONYL COMPOUNDS AS CCR6 INHIBITORS ChemoCentryx, Inc. (US) 2024-06-26 EP disclosed
US-12012403-B2 Aryl sulfonyl compounds as CCR6 inhibitors CHEMOCENTRYX, INC. (US) 2024-06-18 US disclosed
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer INVENTIVA (FR) 2024-06-04 US disclosed
CN-118019735-A Arylsulfonyl compounds as CCR6 inhibitors 坎莫森特里克斯公司 2024-05-10 CN disclosed
CN-113039182-B Inhibitors of YAP/TAZ-TEAD interactions and their use in cancer treatment 伊文蒂瓦公司 2024-02-20 CN disclosed
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed
WO-2010038081-A2 HETEROCYCLIC DERIVATIVES AND METHODS OF USE THEREOF ASTRAZENECA AB (SE) 2010-04-08 WO disclosed
US-7671221-B2 Modulators of ATP-Binding Cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-03-02 US disclosed
US-7671221-B2 Modulators of ATP-Binding Cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-03-02 US disclosed
US-7671221-B2 Modulators of ATP-Binding Cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-03-02 US disclosed
US-20090192154-A1 SULTAM DERIVATIVES ASAHI KASEI PHARMA CORPORATION (JP) 2009-07-30 US disclosed
WO-2009006315-A1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS FOR TREATING CYSTIC FIBROSIS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-01-08 WO disclosed
US-20080009524-A1 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED 2008-01-10 US disclosed
US-20080009524-A1 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED 2008-01-10 US disclosed
US-20080009524-A1 Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED 2008-01-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12012403-B2 Aryl sulfonyl compounds as CCR6 inhibitors CCR6, CCR1, CCR3 CHEK1 1363/4885DAPK3 2657/4885MAP4K4 2953/4885
US-20080009524-A1 Modulators of ATP-binding cassette transporters CFTR, ABCB1, ABCC2 CHEK1 4693/4885DAPK3 4344/4885MAP4K4 4714/4885
US-11999758-B2 Inhibitors of the YAP/TAZ-TEAD interaction and their use in the treatment of cancer YAP1, TEAD2, YES1 CHEK1 125/4885DAPK3 247/4885MAP4K4 469/4885
US-20260092053-A1 KHK INHIBITORS KHK, SLC5A2, HK1 CHEK1 2740/4885DAPK3 3216/4885MAP4K4 227/4885
US-20090192154-A1 SULTAM DERIVATIVES SULT1A1, SULT2A1, ADAMTS1 CHEK1 4647/4885DAPK3 4519/4885MAP4K4 4513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.