SCHEMBL1701666

SCHEMBL1701666

CC(=O)Oc1cc(C)cc(OC(C)=O)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.63
MAPT P10636 4/20 0.52
KDM4E B2RXH2 4/20 0.52
CYP3A4 P08684 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TTR P02766 1/20 0.52
TP53 P04637 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ELANE P08246 2/20 0.51
CYP19A1 P11511 1/20 0.47
ACHE P22303 2/20 0.46
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
BACE1 P56817 1/20 0.46
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
HSD17B10 Q99714 2/20 0.42
GLA P06280 2/20 0.42
GAA P10253 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593772 0.95 LMNA (0.63) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL28793573 0.93 LMNA (0.61) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL14707645 0.91 LMNA (0.55) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL2010436 0.89 LMNA (0.59) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL17188986 0.89 LMNA (0.53) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL10149317 0.88 LMNA (0.52) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL6749439 0.87 LMNA (0.55) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL10149312 0.86 LMNA (0.69) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL16957540 0.86 LMNA (0.50) LMNAMAPTKDM4ECYP3A4MEN1
SCHEMBL16950528 0.86 LMNA (0.55) LMNAMAPTKDM4ECYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193789-B1 The application of 3,5-dihydroxytoluene or derivatives thereof in the preparation of medicine and functional food for treating or preventing depression KUNMING INST BOTANY CN ACAD (CN) 2013-02-20 EP claimed
US-20100190730-A1 APPLICATION OF 5-METHYL-1,3-BENZENEDIOL OR DERIVATIVES THEREOF IN THE PREPARATION OF MEDICINES AND FUNCTIONAL FOODS FOR TREATMENT OR PREVENTION OF DEPRESSION KUNMING INSTITUTE OF BOTANY, CHINESE ACADEMY OF SCIENCES (CN) 2010-07-29 US claimed
EP-2193789-A1 THE APPLICATION OF 3, 5-DIHYDROXYTOLUENE OR DERIVATIVES THEREOF IN THE PREPARATION OF MEDICINE AND FUNCTIONAL FOR TREATING OR PREVENTING DEPRESSION. Kunming Institute Of Botany, Chinese Academy Of Sciences (CN) 2010-06-09 EP claimed
WO-2023187302-A1 NOVEL PLASTICIZERS, PROCESS FOR THE PREPARATION THEREOF, AND USE THEREOF ORPIA INNOVATION (FR) 2023-10-05 WO disclosed
US-11583527-B2 Hydantoin derivatives useful as Kv3 inhibitors AUTIFONY THERAPEUTICS LIMITED (GB) 2023-02-21 US disclosed
US-11583527-B2 Hydantoin derivatives useful as Kv3 inhibitors AUTIFONY THERAPEUTICS LIMITED (GB) 2023-02-21 US disclosed
US-20220054490-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS AUTIFONY THERAPEUTICS LIMITED (GB) 2022-02-24 US disclosed
US-20220054490-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS AUTIFONY THERAPEUTICS LIMITED (GB) 2022-02-24 US disclosed
US-11197859-B2 Hydantoin derivatives useful as Kv3 inhibitors AUTIFONY THERAPEUTICS LIMITED (GB) 2021-12-14 US disclosed
US-11136343-B2 Binuclear metal complexes for use as emitters in organic electroluminescent devices MERCK PATENT GMBH (DE) 2021-10-05 US disclosed
US-20200360379-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS GLAXOSMITHKLINE S.P.A. (IT) 2020-11-19 US disclosed
EP-2193789-A1 THE APPLICATION OF 3, 5-DIHYDROXYTOLUENE OR DERIVATIVES THEREOF IN THE PREPARATION OF MEDICINE AND FUNCTIONAL FOR TREATING OR PREVENTING DEPRESSION. Kunming Institute Of Botany, Chinese Academy Of Sciences (CN) 2010-06-09 EP disclosed
EP-2193789-A1 THE APPLICATION OF 3, 5-DIHYDROXYTOLUENE OR DERIVATIVES THEREOF IN THE PREPARATION OF MEDICINE AND FUNCTIONAL FOR TREATING OR PREVENTING DEPRESSION. Kunming Institute Of Botany, Chinese Academy Of Sciences (CN) 2010-06-09 EP disclosed
US-7528140-B2 Substituted pyrrolo[3,2-d]pyrimidines as glycogen synthase kinase (GSK) inhibitors TEIJIN LIMITED (JP) 2009-05-05 US disclosed
US-7528140-B2 Substituted pyrrolo[3,2-d]pyrimidines as glycogen synthase kinase (GSK) inhibitors TEIJIN LIMITED (JP) 2009-05-05 US disclosed
US-7323458-B1 Dihydrobenzodiazepins and their use for treating dyslipidemia MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2008-01-29 US disclosed
US-7323458-B1 Dihydrobenzodiazepins and their use for treating dyslipidemia MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2008-01-29 US disclosed
EP-1663234-A1 PIPERAZINE DERIVATIVES FOR THE TREATMENT OF HIV INFECTIONS Pfizer Limited (GB) 2006-06-07 EP disclosed
US-20050043300-A1 Piperazine derivatives PFIZER INC. 2005-02-24 US disclosed
WO-2005016344-A1 PIPERAZINE DERIVATIVES FOR THE TREATMENT OF HIV INFECTIONS PFIZER LIMITED (GB) 2005-02-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11583527-B2 Hydantoin derivatives useful as Kv3 inhibitors KCNN3, KCND3, KCNA3 LMNA 1917/4885MAPT 3926/4885KDM4E 1460/4885
US-20220054490-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS KCNN3, KCND3, KCNA3 LMNA 1917/4885MAPT 3926/4885KDM4E 1460/4885
US-20200360379-A1 HYDANTOIN DERIVATIVES USEFUL AS KV3 INHIBITORS KCNN3, KCND3, KCNA3 LMNA 1917/4885MAPT 3926/4885KDM4E 1460/4885
US-20050043300-A1 Piperazine derivatives CD4, CCR5, RRP15 LMNA 3961/4885MAPT 2428/4885KDM4E 2439/4885
US-11136343-B2 Binuclear metal complexes for use as emitters in organic electroluminescent devices AP2M1, MCU, AP3M1 LMNA 3190/4885MAPT 1256/4885KDM4E 4613/4885
US-20100190730-A1 APPLICATION OF 5-METHYL-1,3-BENZENEDIOL OR DERIVATIVES THEREOF IN THE PREPARATION OF MEDICINES AND FUNCTIONAL FOODS FOR TREATMENT OR PREVENTION OF DEPRESSION TPH1, TPH2, HTR5A LMNA 597/4885MAPT 3939/4885KDM4E 143/4885
US-11197859-B2 Hydantoin derivatives useful as Kv3 inhibitors KCNN3, KCND3, KCNA3 LMNA 1917/4885MAPT 3926/4885KDM4E 1460/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.