SCHEMBL17023146

SCHEMBL17023146

Cc1cscc1-c1ccc(OC(=O)Nc2ncc[nH]2)c2nccnc12

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.34
ADRA2C P18825 3/20 0.34
PTGES O14684 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
FFAR2 O15552 1/20 0.33
CYP2A6 P11509 3/20 0.33
HSP90AA1 P07900 1/20 0.33
HPGDS O60760 1/20 0.32
NR3C1 P04150 1/20 0.31
FGFR3 P22607 1/20 0.31
CYP2E1 P05181 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2B6 P20813 1/20 0.30
CYP2C19 P33261 1/20 0.30
CHRM4 P08173 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17023184 0.83 HSP90AA1 (0.38) ADRA2AADRA2CPTGESADRA1DADRA1A
SCHEMBL1126185 0.82 PTGES (0.43) ADRA2AADRA2CPTGESHPGDSFGFR3
SCHEMBL17023018 0.79 FGFR3 (0.45) HSP90AA1NR3C1FGFR3CYP2C9
SCHEMBL17023080 0.79 HSP90AA1 (0.38) ADRA2AHSP90AA1NR3C1FGFR3
SCHEMBL17023143 0.77 HSP90AA1 (0.44) ADRA2AADRA2CHSP90AA1FGFR3CYP3A4
SCHEMBL17023037 0.76 HPGDS (0.44) ADRA2AADRA2CPTGESADRA1DADRA1A
SCHEMBL17023104 0.76 FGFR3 (0.53) FGFR3
SCHEMBL17023129 0.75 FGFR3 (0.46) HSP90AA1FGFR3CYP3A4
SCHEMBL17023075 0.71 FGFR3 (0.54) FGFR3
SCHEMBL17023116 0.71 L3MBTL1 (0.48) FGFR3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282995-B1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2015-08-26 EP claimed