SCHEMBL1704439

SCHEMBL1704439

Cc1cc(Nc2cc3ccccc3c(-c3cccc(C4CCN(C(=O)O)CC4)c3)n2)nn1C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MCHR1 Q99705 8/20 0.35
SCD5 Q86SK9 2/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
TPSAB1 Q15661 6/20 0.33
MAP3K12 Q12852 1/20 0.33
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL902875 0.90 IGF1R (0.42)
SCHEMBL902923 0.84 NPC1 (0.36) NPC1RAB9AMCHR1SCD5MAP3K12
SCHEMBL902789 0.81 ALDH1A1 (0.42) NPC1RAB9A
SCHEMBL1705277 0.74 JAK2 (0.44)
SCHEMBL1704146 0.74 NAMPT (0.43)
SCHEMBL902745 0.67 PLK4 (0.44) NPC1RAB9A
SCHEMBL1704634 0.66 ALDH1A1 (0.38) NPC1RAB9A
SCHEMBL901929 0.66 KARS1 (0.55) MAP3K12
SCHEMBL1704967 0.64 ALDH1A1 (0.44) NPC1RAB9AMAP3K12
SCHEMBL901949 0.64 KARS1 (0.48) NPC1RAB9AMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed