SCHEMBL1704967

SCHEMBL1704967

Cc1ccnc(Nc2cc3ccccc3c(-c3cccc(C4=CCN(C(=O)O)CC4)c3)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
MAP3K12 Q12852 6/20 0.43
KDR P35968 2/20 0.41
MAP4K4 O95819 1/20 0.41
ABL1 P00519 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
IGF1R P08069 1/20 0.41
LTK P29376 1/20 0.41
MAP2K2 P36507 1/20 0.41
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
CLK2 P49760 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41
CDK5 Q00535 1/20 0.41
MAP2K1 Q02750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901343 0.89 NAMPT (0.44) CDK9
SCHEMBL1705014 0.88 ALDH1A1 (0.44) ALDH1A1KDM4EKDRCDK9SMN1; SMN2
SCHEMBL902789 0.84 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2KMT2ANPC1
SCHEMBL901312 0.83 KARS1 (0.54) ALDH1A1MAP3K12SMN1; SMN2JAK2KARS1
SCHEMBL901949 0.80 KARS1 (0.48) MAP3K12KDRMAP4K4ABL1LCK
SCHEMBL1705140 0.79 KDR (0.42) MAP3K12KDRMAP4K4ABL1LCK
SCHEMBL901340 0.79 ALDH1A1 (0.50) ALDH1A1KDM4ESMN1; SMN2KMT2ANPC1
SCHEMBL902803 0.78 PDE10A (0.45) CDK9
SCHEMBL1704146 0.75 NAMPT (0.43) ALDH1A1KDM4ECDK7
SCHEMBL901948 0.73 KARS1 (0.46) ALDH1A1KDM4ECDK9SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441755-A1 Pyridine- and isoquinoline-derivatives as Syk and JAK kinase inhibitors Almirall, S.A. (ES) 2012-04-18 EP disclosed