SCHEMBL17079604

SCHEMBL17079604

Cc1ccccc1NC(=O)Nc1cccnc1

nearest known ligand 0.74

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.74
KMT2A Q03164 4/20 0.74
MAPT P10636 2/20 0.74
LMNA P02545 1/20 0.74
ATM Q13315 1/20 0.74
HTT P42858 2/20 0.69
AHR P35869 1/20 0.68
KDM4E B2RXH2 2/20 0.67
HSD17B10 Q99714 1/20 0.67
NOTUM Q6P988 1/20 0.67
NPC1 O15118 3/20 0.66
RAB9A P51151 3/20 0.66
DDX3X O00571 2/20 0.65
IMPDH2 P12268 1/20 0.64
TSHR P16473 1/20 0.58
ALDH1A1 P00352 1/20 0.57
CYP1A2 P05177 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30051982 0.83 MEN1 (0.77) MEN1KMT2AMAPTLMNAATM
SCHEMBL9637653 0.83 MEN1 (0.77) MEN1KMT2AMAPTLMNAATM
SCHEMBL8016258 0.83 NPC1 (0.68) MEN1KMT2AMAPTLMNAATM
SCHEMBL5950228 0.82 HTT (0.66) MEN1KMT2AMAPTLMNAATM
SCHEMBL812756 0.82 DDX3X (0.80) MEN1KMT2AMAPTLMNAHTT
SCHEMBL10665495 0.82 RAB9A (0.79) MEN1KMT2AMAPTLMNAHTT
SCHEMBL824577 0.82 KMT2A (0.69) MEN1KMT2AMAPTLMNAATM
SCHEMBL22926342 0.82 HTT (1.00) MEN1KMT2AMAPTLMNAATM
Bromide SCHEMBL29417998 0.82 MEN1 (0.74) MEN1KMT2AMAPTLMNAATM
Hydrochloric Acid SCHEMBL29388210 0.82 MEN1 (0.74) MEN1KMT2AMAPTLMNAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015136292-A9 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2022-04-21 WO disclosed
WO-2015136292-A9 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2022-04-21 WO disclosed
US-20210022340-A1 USE OF PYRIDINE UREA COMPOUND HAVING SNAIL-KILLING ACTIVITY THE NATIONAL INSTITUTE OF PARASITIC DISEASES, CHINESE CENTER FOR DISEASE CONTROL AND PREVENTION (CN) 2021-01-28 US disclosed
US-9884812-B2 Use of DDX3X inhibitors for the treatment of pneumovirus infections UNIVERSITY OF WARWICK (GB) 2018-02-06 US disclosed
US-9884812-B2 Use of DDX3X inhibitors for the treatment of pneumovirus infections UNIVERSITY OF WARWICK (GB) 2018-02-06 US disclosed
US-20170166519-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2017-06-15 US disclosed
US-20170166519-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2017-06-15 US disclosed
EP-3116852-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS University of Warwick (GB) 2017-01-18 EP disclosed
WO-2015136292-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2015-09-17 WO disclosed
WO-2015136292-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS UNIVERSITY OF WARWICK (GB) 2015-09-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210022340-A1 USE OF PYRIDINE UREA COMPOUND HAVING SNAIL-KILLING ACTIVITY SLC14A1, UACA, UROD MEN1 3057/4885KMT2A 4029/4885MAPT 2676/4885
US-20170166519-A1 USE OF DDX3X INHIBITORS FOR THE TREATMENT OF PNEUMOVIRUS INFECTIONS DDX3X, DDX1, DDX5 MEN1 2244/4885KMT2A 2069/4885MAPT 3569/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.