SCHEMBL1709234

SCHEMBL1709234

c1ccc(CN2CCC3(CC2)CC3CNc2cccc3cccnc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.60
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
RECQL P46063 1/20 0.47
NAMPT P43490 3/20 0.46
GLO1 Q04760 3/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ROCK2 O75116 2/20 0.40
ROCK1 Q13464 1/20 0.40
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR1A P08908 1/20 0.39
HTR2C P28335 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709247 0.76 SCN9A (0.64) SCN9AMEN1KMT2ACYP3A4CYP2D6
SCHEMBL1709232 0.75 SCN9A (1.00) SCN9AMEN1KMT2ACYP3A4NAMPT
SCHEMBL10072406 0.73 SCN9A (0.57) SCN9AMEN1KMT2ACYP3A4CYP2C19
SCHEMBL10071963 0.72 SCN9A (0.56) SCN9AMEN1KMT2ACYP3A4NAMPT
SCHEMBL1709211 0.72 SCN9A (0.59) SCN9AMEN1KMT2ANAMPTHTT
SCHEMBL1709213 0.71 SCN9A (0.58) SCN9ACYP3A4NAMPTKDM4EALDH1A1
SCHEMBL10071962 0.70 SCN9A (0.57) SCN9ACYP3A4NAMPTACHEBACE1
SCHEMBL8053546 0.69 HDAC6 (0.64) MEN1KMT2ARECQLGLO1HTT
SCHEMBL18753515 0.67 NPC1 (0.51) MEN1KMT2AMAPK1HTTSMN1; SMN2
SCHEMBL6637562 0.67 DRD2 (0.61) MEN1KMT2ACYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed