SCHEMBL1709471

SCHEMBL1709471

COC(=O)C[C@@H]1CCCC(=O)[C@H]1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36
P2RX7 Q99572 1/20 0.35
F2R P25116 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
LMNA P02545 1/20 0.35
MDM2 Q00987 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709470 0.96 KDM4E (0.40) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL1709479 0.88 SLC6A3 (0.36) TDP1
SCHEMBL4549803 0.77 TACR1 (0.41) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL27763781 0.77 ACHE (0.42) LMNA
SCHEMBL1709428 0.75 CYP11B1 (0.43) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL3580847 0.74 TACR1 (0.44) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL1709392 0.73 MAOA (0.44) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL14984450 0.73 DGAT1 (0.47) KDM4EALDH1A1POLBGAAMAPK1
SCHEMBL1709386 0.71 MAOA (0.48)
SCHEMBL8152875 0.71 KDM4E (0.39) KDM4EALDH1A1POLBGAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed